SCHEMBL3720809

SCHEMBL3720809

NC(=O)c1cc(-c2ccc(C(F)(F)F)cc2)nc(N2CCN(Cc3ccc4c(c3)OCO4)CC2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HSD17B10 Q99714 3/20 0.50
PMP22 Q01453 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
USP2 O75604 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
HTR1A P08908 1/20 0.48
ADRA2A P08913 1/20 0.48
CYP2D6 P10635 1/20 0.48
DRD2 P14416 1/20 0.48
ADRA2B P18089 1/20 0.48
ADRA2C P18825 1/20 0.48
NFKB1 P19838 1/20 0.48
SLC6A2 P23975 1/20 0.48
MAPK1 P28482 1/20 0.48
SLC6A4 P31645 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720812 0.85 LMNA (0.59) LMNASMN1; SMN2HSD17B10PMP22MEN1
SCHEMBL3727012 0.85 PARP1 (0.51) LMNASMN1; SMN2HSD17B10USP2CYP3A4
SCHEMBL3717048 0.81 KDM4E (0.52) LMNAHSD17B10PARP1PARP2ALDH1A1
SCHEMBL3797911 0.80 KDM4E (0.56) LMNAHSD17B10MEN1KMT2APARP1
SCHEMBL3717692 0.80 KDM4E (0.55) LMNAHSD17B10PARP1PARP2ALDH1A1
SCHEMBL3721797 0.80 KDM4E (0.52) LMNASMN1; SMN2HSD17B10PARP1PARP2
SCHEMBL3721070 0.78 KDM4E (0.53) LMNAHSD17B10PARP1PARP2ALDH1A1
SCHEMBL3717027 0.78 KDM4E (0.52) LMNAHSD17B10ALDH1A1KDM4EHTT
SCHEMBL3717909 0.78 KDM4E (0.49) LMNAHSD17B10ALDH1A1KDM4EHTT
SCHEMBL3724662 0.77 KDM4E (0.73) LMNASMN1; SMN2HSD17B10MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed