SCHEMBL3721771

SCHEMBL3721771

O=C1CNc2ccc(=O)n3c2N1CCC3CN1CCC(NCc2ccc3c(c2)OCCO3)CC1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.39
TOP2A P11388 1/20 0.36
SLC2A1 P11166 3/20 0.35
MCHR1 Q99705 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL910629 0.99 KCNH2 (0.39) KCNH2TOP2ASLC2A1MCHR1SMN1; SMN2
Hydrochloric Acid SCHEMBL910544 0.99 KCNH2 (0.39) KCNH2TOP2ASLC2A1MCHR1SMN1; SMN2
SCHEMBL910317 0.88 KCNH2 (0.39) KCNH2TOP2A
SCHEMBL3727967 0.88 KCNH2 (0.39) KCNH2TOP2A
Hydrochloric Acid SCHEMBL3731742 0.87 KCNH2 (0.39) KCNH2TOP2A
Hydrochloric Acid SCHEMBL910464 0.87 KCNH2 (0.39) KCNH2TOP2A
SCHEMBL909985 0.86 KCNH2 (0.49) KCNH2TOP2ASLC2A1
SCHEMBL910083 0.86 KCNH2 (0.35) KCNH2TOP2ASLC2A1
Hydrochloric Acid SCHEMBL910352 0.86 KCNH2 (0.49) KCNH2TOP2ASLC2A1
Hydrochloric Acid SCHEMBL910105 0.86 KCNH2 (0.35) KCNH2TOP2ASLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238138-A1 TRICYCLIC NITROGEN COMPOUNDS AND THEIR USE AS ANTIBACTERIAL AGENTS Glaxo Group Limited (GB) 2010-10-13 EP claimed
WO-2009087153-A1 TRICYCLIC NITROGEN COMPOUNDS AND THEIR USE AS ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2009-07-16 WO claimed