SCHEMBL3722007

SCHEMBL3722007

NCc1cc(-c2ccc3c(c2)OCO3)nc(NCc2cccnc2)n1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 12/20 0.71
DYRK1A Q13627 9/20 0.71
CLK1 P49759 8/20 0.71
CLK2 P49760 5/20 0.71
DYRK1B Q9Y463 5/20 0.71
CLK3 P49761 3/20 0.71
CDK2 P24941 1/20 0.71
ALDH1A1 P00352 7/20 0.61
KDM4E B2RXH2 6/20 0.61
HSD17B10 Q99714 5/20 0.61
CYP1A2 P05177 4/20 0.61
CYP3A4 P08684 4/20 0.61
CYP2D6 P10635 4/20 0.61
CYP2C19 P33261 4/20 0.61
CYP2C9 P11712 3/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
ALOX15 P16050 2/20 0.61
MAPK1 P28482 2/20 0.61
HPGD P15428 2/20 0.61
TP53 P04637 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723029 0.81 KDM4E (0.53) CLK4DYRK1ACLK1CLK2DYRK1B
SCHEMBL3718626 0.78 KDM4E (0.61) CDK2ALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL3723229 0.78 ADORA1 (0.48) CLK4DYRK1ACLK1CLK2DYRK1B
SCHEMBL3719658 0.77 DYRK1A (0.49) CLK4DYRK1ACLK1CLK2DYRK1B
SCHEMBL3721197 0.77 ADORA1 (0.51) CLK4DYRK1ACLK1CLK2DYRK1B
SCHEMBL1076858 0.75 CLK4 (0.67) CLK4DYRK1ACLK1CLK2DYRK1B
SCHEMBL3725579 0.74 DYRK1A (0.65) CLK4DYRK1ACLK1CLK2DYRK1B
SCHEMBL3717907 0.74 CLK4 (0.52) CLK4DYRK1ACLK1CLK2DYRK1B
SCHEMBL3724659 0.74 DYRK1A (0.51) CLK4DYRK1ACLK1CLK2DYRK1B
SCHEMBL30250542 0.74 CLK4 (1.00) CLK4DYRK1ACLK1CLK2DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed