SCHEMBL3722156

SCHEMBL3722156

CN1CCCN(c2nc(C(N)=O)cc(-c3ccc(C(F)(F)F)cc3)n2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.67
HTT P42858 2/20 0.67
GLA P06280 1/20 0.67
ALDH1A1 P00352 2/20 0.58
GAA P10253 2/20 0.58
HPGD P15428 2/20 0.58
TP53 P04637 1/20 0.58
HSD17B10 Q99714 2/20 0.57
TSHR P16473 1/20 0.57
CASP1 P29466 1/20 0.57
CASP7 P55210 1/20 0.57
HRH4 Q9H3N8 1/20 0.51
SCN9A Q15858 8/20 0.50
LMNA P02545 1/20 0.50
POLB P06746 1/20 0.50
GPR55 Q9Y2T6 1/20 0.50
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724662 0.96 KDM4E (0.73) KDM4EHTTGLAALDH1A1GAA
SCHEMBL1734132 0.89 KDM4E (0.72) KDM4EHTTGLAALDH1A1GAA
SCHEMBL3728035 0.86 KDM4E (0.71) KDM4EHTTGLAALDH1A1GAA
SCHEMBL3718061 0.84 KDM4E (0.56) KDM4EHTTGLAALDH1A1GAA
SCHEMBL3797911 0.84 KDM4E (0.56) KDM4EHTTGLAALDH1A1GAA
SCHEMBL3726430 0.84 KDM4E (0.57) KDM4EHTTGLAALDH1A1GAA
SCHEMBL3720929 0.83 KDM4E (0.56) KDM4EHTTGLAALDH1A1GAA
SCHEMBL3725417 0.82 SCN9A (0.54) KDM4EHTTGLAALDH1A1GAA
SCHEMBL3724010 0.82 KDM4E (0.54) KDM4EHTTGLAALDH1A1GAA
SCHEMBL3720439 0.82 KDM4E (0.53) KDM4EHTTGLAALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed