SCHEMBL3728035

SCHEMBL3728035

CN1CCCN(c2nc(C(N)=O)cc(-c3ccc(Br)cc3)n2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.71
HTT P42858 2/20 0.71
GLA P06280 1/20 0.71
ALDH1A1 P00352 4/20 0.61
HPGD P15428 3/20 0.61
GAA P10253 2/20 0.61
TP53 P04637 1/20 0.61
HSD17B10 Q99714 2/20 0.61
TSHR P16473 1/20 0.61
CASP1 P29466 1/20 0.61
CASP7 P55210 1/20 0.61
POLB P06746 2/20 0.53
LMNA P02545 1/20 0.53
GPR55 Q9Y2T6 1/20 0.53
HRH4 Q9H3N8 2/20 0.48
HRH3 Q9Y5N1 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 1/20 0.43
CHEK1 O14757 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718071 0.95 KDM4E (0.78) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL3722156 0.86 KDM4E (0.67) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL3719605 0.82 KDM4E (0.58) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL3720910 0.81 LMNA (0.78) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL3724662 0.81 KDM4E (0.73) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL3720247 0.80 SCN9A (0.56) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL3728038 0.80 HRH4 (0.50) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL1733760 0.80 KDM4E (0.92) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL1734353 0.79 KDM4E (0.77) KDM4EHTTGLAALDH1A1HPGD
SCHEMBL3717767 0.78 KDM4E (0.59) KDM4EHTTGLAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed