SCHEMBL3724653

SCHEMBL3724653

CC(=O)c1ccc2nc(Oc3ccc(Nc4ccccc4)cc3)ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.53
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
HSP90AA1 P07900 1/20 0.45
GAA P10253 1/20 0.45
SCD O00767 1/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 2/20 0.44
GLA P06280 1/20 0.44
HTT P42858 2/20 0.44
GUSB P08236 1/20 0.44
AKR1C3 P42330 2/20 0.43
AKR1C2 P52895 2/20 0.43
PIN1 Q13526 2/20 0.42
MCHR1 Q99705 1/20 0.40
PLAU P00749 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721861 0.83 PDE4B (0.53) PDE4BALDH1A1MAPTGAANPC1
SCHEMBL3720024 0.83 PDE4B (0.53) PDE4BALDH1A1MAPTGAANPC1
SCHEMBL3717735 0.81 PDE4B (0.57) PDE4BALDH1A1MAPTGAASCD
SCHEMBL13076364 0.80 ACACB (0.50)
SCHEMBL3722547 0.80 PDE4B (0.52) PDE4BMAPTNPC1RAB9AKMT2A
SCHEMBL3724294 0.79 PDE4B (0.55) PDE4BALDH1A1MAPTGAARAB9A
SCHEMBL3723898 0.78 PDE4B (0.50) PDE4BMAPTGAANPC1RAB9A
SCHEMBL3721431 0.78 PDE4B (0.53) PDE4BALDH1A1LMNAGLAAKR1C3
SCHEMBL3718630 0.78 PDE4B (0.54) PDE4BALDH1A1MAPT
SCHEMBL3717019 0.78 CYP1A2 (0.43) ALDH1A1MAPTNPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed