SCHEMBL3717019

SCHEMBL3717019

CCc1ccc2nc(Oc3ccc(Nc4ccccc4)cc3)ccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
CYP2A6 P11509 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
FGFR2 P21802 1/20 0.39
RAB9A P51151 3/20 0.39
NPC1 O15118 1/20 0.39
MAPKAPK2 P49137 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
RAD52 P43351 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719857 0.85 ALDH1A1 (0.37) ALDH1A1CYP3A4HPGDHSD17B10FGFR2
SCHEMBL3725263 0.85 MAPT (0.42) CYP1A2CYP2A6SMN1; SMN2MAPTALDH1A1
SCHEMBL3720909 0.82 RAB9A (0.39) CYP1A2CYP2A6SMN1; SMN2MAPTALDH1A1
SCHEMBL3720524 0.82 SMN1; SMN2 (0.39) CYP1A2CYP2A6SMN1; SMN2MAPTALDH1A1
SCHEMBL3716766 0.81 SMN1; SMN2 (0.43) CYP1A2CYP2A6SMN1; SMN2MAPTTP53
SCHEMBL3722368 0.81 HTT (0.52) CYP1A2SMN1; SMN2MAPTALDH1A1HPGD
SCHEMBL3722417 0.79 MEN1 (0.38) SMN1; SMN2MAPTALDH1A1HSD17B10FGFR2
SCHEMBL3724653 0.78 PDE4B (0.53) MAPTALDH1A1RAB9ANPC1KMT2A
SCHEMBL3719854 0.78 FGFR2 (0.37) SMN1; SMN2MAPTALDH1A1CYP3A4HPGD
SCHEMBL18236258 0.77 CYP1A2 (0.47) CYP1A2CYP2A6SMN1; SMN2MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO claimed
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed