SCHEMBL3724911

SCHEMBL3724911

Cc1cc(C2CC(N)CCN2C(=O)OC(C)(C)C)c2[nH]c(-c3ccccc3)cc2c1.Cc1cc(NC2CCNCC2)c2[nH]c(-c3ccccc3)cc2c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.38
BRD4 O60885 5/20 0.35
ATAD2 Q6PL18 4/20 0.35
VCP P55072 2/20 0.34
CHEK1 O14757 1/20 0.33
KCNH2 Q12809 1/20 0.33
BACE1 P56817 1/20 0.33
KHK P50053 1/20 0.32
LMNA P02545 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PIM1 P11309 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
GAA P10253 1/20 0.31
TSHR P16473 1/20 0.31
USP30 Q70CQ3 1/20 0.31
NR1H2 P55055 2/20 0.31
NR1H3 Q13133 1/20 0.30
HPGDS O60760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2995214 0.89 KIT (0.42) KITVCPBACE1LMNANPSR1
SCHEMBL3723438 0.86 KIT (0.39) KITVCPLMNANPSR1TSHR
SCHEMBL3724914 0.84 KIT (0.48) KITBRD4VCPBACE1PIM1
SCHEMBL2995216 0.80 KIT (0.52) KITBRD4VCPBACE1PIM1
SCHEMBL3723439 0.77 KIT (0.49) KITBRD4VCPBACE1PIM1
SCHEMBL2999762 0.77 BRD4 (0.48) BRD4ATAD2CHEK1KCNH2KHK
Hydrochloric Acid SCHEMBL3415428 0.76 BRD4 (0.47) BRD4ATAD2CHEK1KCNH2KHK
SCHEMBL3109553 0.72 NPY5R (0.44) BRD4ATAD2CHEK1KCNH2KHK
SCHEMBL3000216 0.71 NPY5R (0.50) BRD4CHEK1KCNH2BACE1PIM1
SCHEMBL3005991 0.69 CHEK1 (0.40) VCPCHEK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2178870-A1 INDOLE AND INDAZOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG Life Sciences Ltd. (KR) 2010-04-28 EP disclosed
WO-2009025478-A1 INDOLE AND INDAZOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG LIFE SCIENCES LTD. (KR) 2009-02-26 WO disclosed