SCHEMBL3725632

SCHEMBL3725632

Cc1c(N)cccc1OCCN1CCOCC1

nearest known ligand 0.75

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.64
POLB P06746 2/20 0.56
DRD1 P21728 1/20 0.53
DRD4 P21917 1/20 0.53
DRD5 P21918 1/20 0.53
TSHR P16473 2/20 0.52
CYP2D6 P10635 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
HTR1A P08908 1/20 0.51
KDM4E B2RXH2 3/20 0.50
SYK P43405 1/20 0.49
P2RY12 Q9H244 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5463193 0.87 TDP1 (0.63) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL30726450 0.86 DRD1 (0.56) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL1853220 0.85 DRD1 (0.62) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL13744516 0.84 SMN1; SMN2 (0.66) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL2011534 0.84 CYP2D6 (0.60) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL25374902 0.83 KDM4E (0.57) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL28937449 0.83 POLB (0.64) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL29559230 0.83 POLB (0.64) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL1953267 0.83 TSHR (0.56) SMN1; SMN2POLBDRD1DRD4DRD5
SCHEMBL5235337 0.82 DRD1 (0.52) SMN1; SMN2POLBDRD1DRD4DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125103-A1 DIKETOPIPERAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2010-11-04 WO disclosed