SCHEMBL3728010

SCHEMBL3728010

CN1CCN(c2ccc(-c3cccc(CN)c3)cc2)CC1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 6/20 0.66
AGXT P21549 1/20 0.50
CHKA P35790 1/20 0.49
JAK2 O60674 1/20 0.48
CTSK P43235 4/20 0.47
CTSL P07711 3/20 0.47
ADRA2C P18825 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
GFER P55789 1/20 0.47
KMT2A Q03164 1/20 0.47
PTK2B Q14289 1/20 0.47
ESR2 Q92731 1/20 0.47
ASIC3 Q9UHC3 1/20 0.47
MELK Q14680 1/20 0.45
CTSB P07858 2/20 0.43
CTSS P25774 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721910 0.85 CHKA (0.57) AOC3AGXTCHKAKDM4EALDH1A1
SCHEMBL3722035 0.84 AOC3 (0.62) AOC3AGXTCHKAADRA2CALDH1A1
SCHEMBL109344 0.83 AGXT (0.69) AOC3AGXTCHKAADRA2CKDM4E
SCHEMBL111714 0.82 GAA (0.62) AOC3AGXTCHKAADRA2CKDM4E
SCHEMBL12547524 0.81 AOC3 (0.46) AOC3AGXTADRA2C
SCHEMBL12812550 0.80 AOC3 (0.76) AOC3
SCHEMBL14290769 0.80 AOC3 (0.63) AOC3CTSKCTSLMAPTCTSB
SCHEMBL11359440 0.80 AOC3 (1.00) AOC3
SCHEMBL28845811 0.80 ADRA2C (0.70) AOC3AGXTJAK2ADRA2CKDM4E
SCHEMBL29789664 0.80 CHKA (0.56) AOC3CHKAJAK2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed