SCHEMBL3733246

SCHEMBL3733246

Cc1ncn(Cc2ccccc2CC(=O)O)c1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.54
AKR1B1 P15121 1/20 0.42
PTGDR2 Q9Y5Y4 8/20 0.41
KDM4E B2RXH2 3/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
FDPS P14324 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
KMT2A Q03164 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726218 0.73 CYP19A1 (0.54) CYP19A1AKR1B1PTGDR2KDM4ECYP1A2
Iodide SCHEMBL31305035 0.73 AKR1B1 (0.73) CYP19A1AKR1B1KDM4ECYP1A2MAPT
Methyl Alcohol SCHEMBL28299530 0.71 AKR1B1 (0.70) CYP19A1AKR1B1KDM4ECYP1A2MAPT
SCHEMBL30359 0.71 AKR1B1 (0.76) AKR1B1KDM4ECYP1A2MAPTHPGD
SCHEMBL29410826 0.71 AKR1B1 (0.76) AKR1B1KDM4ECYP1A2MAPTHPGD
SCHEMBL3736357 0.71 CYP19A1 (0.48) CYP19A1AKR1B1PTGDR2KDM4ECYP1A2
SCHEMBL3736113 0.70 CYP19A1 (0.48) CYP19A1AKR1B1PTGDR2KDM4ECYP11B1
SCHEMBL28842838 0.69 AKR1B1 (0.73) AKR1B1KDM4ECYP1A2MAPTHPGD
Hydrochloric Acid SCHEMBL6767821 0.69 AKR1B1 (0.73) AKR1B1KDM4ECYP1A2MAPTHPGD
Hydrogen Sulfide SCHEMBL27426416 0.69 AKR1B1 (0.73) AKR1B1KDM4ECYP1A2MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010142652-A1 IMIDAZOBENZAZEPINE COMPOUNDS FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM (CNS) DISEASES GLAXO GROUP LIMITED (GB) 2010-12-16 WO disclosed