SCHEMBL3736658

SCHEMBL3736658

CCOC(=O)c1[nH]ccc1/N=C\N(C)C

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.49
HSD17B10 Q99714 2/20 0.49
LMNA P02545 2/20 0.49
MAPK1 P28482 1/20 0.44
HTT P42858 3/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 2/20 0.44
PKM P14618 1/20 0.42
TSHR P16473 1/20 0.41
KDM4E B2RXH2 7/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
KMT2A Q03164 3/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NUDT1 P36639 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13560529 1.00 ALDH1A1 (0.49) ALDH1A1HSD17B10LMNAMAPK1HTT
SCHEMBL29211279 0.78 KDM4E (0.36) ALDH1A1HSD17B10LMNAMAPK1HTT
SCHEMBL31575794 0.78 KMT2A (0.46) ALDH1A1HSD17B10LMNAMAPK1HTT
SCHEMBL951646 0.75 ALDH1A1 (0.52) ALDH1A1HSD17B10LMNAMAPK1HTT
SCHEMBL2564768 0.74 GRM6 (0.41) ALDH1A1GAAMAPTTSHRKDM4E
SCHEMBL3641814 0.74 KDM4E (0.52) ALDH1A1HSD17B10LMNAMAPK1HTT
SCHEMBL13560604 0.74 KDM4E (0.52) ALDH1A1HSD17B10LMNAMAPK1HTT
SCHEMBL6182362 0.73 TSHR (0.46) ALDH1A1HSD17B10LMNAMAPK1HTT
SCHEMBL6182359 0.73 TSHR (0.46) ALDH1A1HSD17B10LMNAMAPK1HTT
SCHEMBL1149707 0.72 KDM4E (0.47) ALDH1A1LMNAGAATSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304419-B2 Chemical compounds GLAXOSMITHKLINE LLC (US) 2012-11-06 US disclosed
EP-2166856-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2010-03-31 EP disclosed
WO-2008154271-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-18 WO disclosed