Phenylalanine

Phenylalanine

SCHEMBL37367

C[C@H](N)C(=O)O.N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.85

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 6/20 0.85
ALPI P09923 1/20 0.85
PKM P14618 1/20 0.85
PTGS1 P23219 1/20 0.85
XIAP P98170 1/20 0.85
SLC1A3 P43003 2/20 0.61
SLC1A2 P43004 2/20 0.61
SLC1A1 P43005 2/20 0.61
SLC15A1 P46059 1/20 0.56
NOS3 P29474 1/20 0.55
NOS1 P29475 1/20 0.55
NOS2 P35228 1/20 0.55
SLC6A2 P23975 2/20 0.55
TAAR1 Q96RJ0 2/20 0.55
MAOA P21397 1/20 0.55
SLC6A4 P31645 1/20 0.55
SLC6A3 Q01959 1/20 0.55
SIGMAR1 Q99720 1/20 0.55
CYP2A6 P11509 1/20 0.55
ADORA2A P29274 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenylalanine SCHEMBL9226754 1.00 SLC7A5 (0.85) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL28229442 1.00 SLC7A5 (0.85) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL6535507 1.00 SLC7A5 (0.85) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL8910300 1.00 SLC7A5 (0.85) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL3486837 1.00 SLC7A5 (0.85) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL2063249 1.00 SLC7A5 (0.85) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL6033327 1.00 SLC7A5 (0.85) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL28667668 0.93 SLC7A5 (0.73) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL3057091 0.93 SLC7A5 (0.73) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL17103846 0.93 SLC7A5 (0.73) SLC7A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2811 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240239885-A1 ANTIBODY CONJUGATE COMPRISING ANTI-P-CADHERIN ANTIBODY AND USES THEREOF WuXi Biologics Ireland Limited (IE) 2024-07-18 US claimed
WO-2023195805-A9 ITGB2-MEDIATED DRUG DELIVERY SYSTEM 트윈피그바이오랩(주) 2024-07-11 WO claimed
WO-2024140917-A1 ANTI-CD40 ANTIBODY-DRUG CONJUGATE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 上海盛迪医药有限公司 2024-07-04 WO claimed
EP-4393515-A1 ANTI-CLDN-18.2 ANTIBODY-DRUG CONJUGATE AND USE THEREOF Shanghai Junshi Biosciences Co., Ltd. (CN) 2024-07-03 EP claimed
CN-118141945-A HER2 nanobody drug conjugates 香港城市大学深圳福田研究院 2024-06-07 CN claimed
US-20240156978-A1 MAYTANSINE-ANTIBODY CONJUGATES AND METHODS OF USING SAME ANGIEX, INC. 2024-05-16 US claimed
CN-117980327-A Specific coupling of antibodies 杭州多禧生物科技有限公司 2024-05-03 CN claimed
EP-4346867-A1 COMPOSITIONS FOR TREATING INFLAMMATORY AIRWAY DISEASE AND USES THEREOF Lateral Pharma Pty Ltd (AU) 2024-04-10 EP claimed
US-11951173-B2 Tetravalent antibody-drug conjugates and use thereof Bliss Biopharmaceutical (Hangzhou) Co., Ltd. (CN) 2024-04-09 US claimed
WO-2024067670-A1 ANTIBODY AND CONJUGATE 苏州智核生物医药科技有限公司 2024-04-04 WO claimed
EP-1718667-A2 HETEROCYCLIC SELF-IMMOLATIVE LINKERS AND CONJUGATES GENENTECH, INC. (US) 2006-11-08 EP claimed
WO-2006078257-A1 SUBSTITUTED FULLERENE COMPOSITIONS AND THEIR USE IN TREATMENT OF SHOCK C SIXTY INC. (US) 2006-07-27 WO claimed
EP-1670718-A2 SUBTITUTED FULLERENE COMPOSITIONS AND THEIR USE AS ANTIOXYDANTS C Sixty Inc. (US) 2006-06-21 EP claimed
US-20050256030-A1 for linking drug moieties to ligands; comprises a peptide sequence that is a substrate for an intracellular enzyme, for example a cathepsin, that cleaves the peptide at an amide bond SEAGEN INC. 2005-11-17 US claimed
WO-2005082023-A2 HETEROCYCLIC SELF-IMMOLATIVE LINKERS AND CONJUGATES GENENTECH, INC. (US) 2005-09-09 WO claimed
WO-2005035441-A2 SUBTITUTED FULLERENE COMPOSITIONS AND THEIR USE AS ANTIOXYDANTS C SIXTY INC. (US) 2005-04-21 WO claimed
EP-1064010-A4 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME CONNECTIVE TISSUE IMAGINEERING (US) 2004-10-06 EP claimed
EP-1064010-A1 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME Mrs, Llc (US) 2001-01-03 EP claimed
WO-1999045941-A1 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME MRS, LLC (US) 1999-09-16 WO claimed
EP-0076557-B1 PEPTIDES AND PSEUDOPEPTIDES IN WHICH THE N TERMINUS BEARS TWO SUBSTITUENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-11-13 EP claimed