SCHEMBL374151

SCHEMBL374151

Cc1ccc(NC(=O)c2ccc(CN3CCN(C)CC3)c(C(F)(F)F)c2)cc1NC(=O)N(C)c1cc(N(C(=O)O)C(C)(C)C)ncn1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRAF P15056 14/20 0.62
EGFR P00533 11/20 0.62
CSF1R P07333 6/20 0.60
KIT P10721 6/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL374394 0.90 BRAF (0.63) BRAFEGFRCSF1RKIT
SCHEMBL374116 0.90 BRAF (0.66) BRAFEGFRCSF1RKIT
SCHEMBL374756 0.88 BRAF (0.63) BRAFEGFRCSF1RKIT
SCHEMBL374244 0.88 BRAF (0.66) BRAFEGFRCSF1RKIT
SCHEMBL374512 0.87 BRAF (0.61) BRAFEGFRCSF1RKIT
SCHEMBL374321 0.87 BRAF (0.70) BRAFEGFRCSF1RKIT
SCHEMBL374349 0.85 BRAF (0.67) BRAFEGFRCSF1RKIT
SCHEMBL374363 0.84 BRAF (0.65) BRAFEGFRCSF1RKIT
SCHEMBL374152 0.82 BRAF (0.42) BRAFEGFRCSF1RKIT
SCHEMBL15121678 0.82 BRAF (0.56) BRAFEGFRCSF1RKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2409969-A1 Pyrimidine urea derivatives as kinase inhibitors Novartis AG (CH) 2012-01-25 EP disclosed