SCHEMBL374152

SCHEMBL374152

Cc1ccc(NC(=O)c2c(F)c(C)c(CN3CCN(C)CC3)c(F)c2F)cc1NC(=O)N(C)c1cc(N(C(=O)O)C(C)(C)C)ncn1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRAF P15056 15/20 0.42
EGFR P00533 12/20 0.42
KIT P10721 5/20 0.40
CSF1R P07333 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL374395 0.89 FGFR3 (0.44) BRAFEGFRKIT
SCHEMBL374151 0.82 BRAF (0.62) BRAFEGFRKITCSF1R
SCHEMBL374384 0.76 FGFR3 (0.60) BRAFEGFRKIT
SCHEMBL374394 0.72 BRAF (0.63) BRAFEGFRKITCSF1R
SCHEMBL374116 0.71 BRAF (0.66) BRAFEGFRKITCSF1R
SCHEMBL15121678 0.71 BRAF (0.56) BRAFEGFRKITCSF1R
SCHEMBL374756 0.70 BRAF (0.63) BRAFEGFRKITCSF1R
SCHEMBL374244 0.70 BRAF (0.66) BRAFEGFRKITCSF1R
SCHEMBL374321 0.70 BRAF (0.70) BRAFEGFRKITCSF1R
SCHEMBL374512 0.69 BRAF (0.61) BRAFEGFRKITCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2409969-A1 Pyrimidine urea derivatives as kinase inhibitors Novartis AG (CH) 2012-01-25 EP disclosed