SCHEMBL3751527

SCHEMBL3751527

[CH2]Oc1ccc(Cl)c2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.59
CYP2A6 P11509 3/20 0.59
TSHR P16473 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
TDP1 Q9NUW8 3/20 0.47
NPSR1 Q6W5P4 1/20 0.47
LMNA P02545 3/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
GPR84 Q9NQS5 6/20 0.41
ESRRA P11474 2/20 0.41
MAPK1 P28482 1/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9188264 0.77 CYP1A2 (0.59) CYP1A2CYP2A6TSHRNPC1RAB9A
SCHEMBL5099452 0.77 CYP1A2 (0.59) CYP1A2CYP2A6TSHRNPC1RAB9A
SCHEMBL29494605 0.77 CYP2A6 (1.00) CYP1A2CYP2A6TSHRNPC1RAB9A
SCHEMBL2473555 0.77 CYP2A6 (1.00) CYP1A2CYP2A6TSHRNPC1RAB9A
SCHEMBL9066455 0.77 CYP1A2 (0.52) CYP1A2CYP2A6TSHRNPC1RAB9A
SCHEMBL29100409 0.76 CYP1A2 (0.56) CYP1A2CYP2A6TSHRNPC1RAB9A
SCHEMBL2091118 0.74 IDO1 (0.59) CYP1A2LMNAKMT2AALDH1A1MAPT
SCHEMBL13019803 0.74 CYP1A2 (0.54) CYP1A2CYP2A6TSHRNPC1RAB9A
SCHEMBL13391184 0.72 CYP1A2 (0.52) CYP1A2CYP2A6TSHRNPC1RAB9A
SCHEMBL29112050 0.72 TSHR (0.53) CYP1A2CYP2A6TSHRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8426631-B2 Fungicidal compounds, method for the production thereof, and use thereof to combat damaging fungi, and agents comprising the same BASF SE (DE) 2013-04-23 US disclosed
US-20100304966-A1 Fungicidal Compounds, Method For the Production Thereof, And Use Thereof To Combat Damaging Fungi, And Agents Comprising The Same BASF SE (DE) 2010-12-02 US disclosed
US-7365082-B2 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines BAYER CROPSCIENCE AG (DE) 2008-04-29 US disclosed
EP-1572668-A4 N-(SUBSTITUTED ARYLMETHYL)-4-(DISUBSTITUTED METHYL)PIPERIDINES AND PIPERAZINES FMC CORP (US) 2006-12-06 EP disclosed
US-20060166962-A1 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines FMC CORPORATION 2006-07-27 US disclosed
EP-1572668-A2 N-(SUBSTITUTED ARYLMETHYL)-4-(DISUBSTITUTED METHYL)PIPERIDINES AND PIPERAZINES FMC CORPORATION (US) 2005-09-14 EP disclosed
WO-2004060865-A2 N-(SUBSTITUTED ARYLMETHYL)-4-(DISUBSTITUTED METHYL)PIPERIDINES AND PIPERAZINES FMC CORPORATION (US) 2004-07-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060166962-A1 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines DDT, DRD4, DRD1 CYP1A2 927/4885CYP2A6 1697/4885TSHR 1446/4885
US-20100304966-A1 Fungicidal Compounds, Method For the Production Thereof, And Use Thereof To Combat Damaging Fungi, And Agents Comprising The Same CYP51A1, ERG28, CAT CYP1A2 22/4885CYP2A6 279/4885TSHR 4645/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.