Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL3752555

COc1ccc2c(c1)c(CC(=O)N(C)C1CCN(C)CC1)cn2S(=O)(=O)c1ccc(Br)s1.O=C(O)C(F)(F)F

nearest known ligand 0.45

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Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 17/20 0.45
CYP3A4 P08684 4/20 0.42
CYP2D6 P10635 4/20 0.42
ADRA2A P08913 2/20 0.42
ADRA2C P18825 2/20 0.42
CYP2C19 P33261 2/20 0.42
HTR2A P28223 1/20 0.42
PPARG P37231 3/20 0.41
PPARD Q03181 3/20 0.41
PPARA Q07869 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3761902 0.88 HTR6 (0.40) HTR6CYP3A4CYP2D6ADRA2AADRA2C
SCHEMBL3752558 0.80 HTR6 (0.37) HTR6CYP3A4CYP2D6ADRA2AADRA2C
Trifluoroacetic Acid SCHEMBL3748726 0.78 HTR6 (0.39) HTR6CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL3744507 0.75 HTR6 (0.39) HTR6
Trifluoroacetic Acid SCHEMBL3749336 0.72 HTR6 (0.39) HTR6
SCHEMBL14572432 0.71 PPARG (0.55) HTR6PPARGPPARDPPARA
Trifluoroacetic Acid SCHEMBL3759250 0.70 HTR6 (0.49) HTR6CYP3A4CYP2D6ADRA2AADRA2C
Trifluoroacetic Acid SCHEMBL3750563 0.68 HTR6 (0.38) HTR6
SCHEMBL5660874 0.67 PPARG (0.61) HTR6PPARGPPARDPPARA
SCHEMBL4605024 0.67 PPARD (0.61) HTR6PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7838518-B2 1-arylsulfonyl-3-substituted indole and indoline derivatives useful in the treatment of central nervous system disorders N.V. ORGANON (NL) 2010-11-23 US disclosed