SCHEMBL375623

SCHEMBL375623

FC(F)(F)Oc1cc(Cl)cc(CNC2CCOCC2)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.46
ACHE P22303 2/20 0.46
BACE1 P56817 2/20 0.46
CARM1 Q86X55 2/20 0.44
PRMT6 Q96LA8 2/20 0.44
EPAS1 Q99814 1/20 0.42
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
OPRL1 P41146 4/20 0.37
FFAR4 Q5NUL3 2/20 0.37
SCN9A Q15858 2/20 0.37
DDR1 Q08345 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
POLB P06746 1/20 0.35
MAP4K4 O95819 1/20 0.34
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL375144 0.82 POLB (0.46) BCHEACHEBACE1CARM1PRMT6
SCHEMBL375222 0.81 CARM1 (0.61) BCHEACHEBACE1CARM1PRMT6
SCHEMBL374832 0.80 BCHE (0.60) BCHEACHEBACE1CARM1PRMT6
SCHEMBL375548 0.76 EPHX1 (0.45) BCHEACHEBACE1CARM1PRMT6
SCHEMBL375224 0.74 OPRL1 (0.42) BCHEACHEBACE1CARM1PRMT6
SCHEMBL375509 0.74 PARP1 (0.44) BCHEACHEBACE1CARM1PRMT6
SCHEMBL374836 0.71 CARM1 (0.51) CARM1PRMT6OPRL1SCN9A
SCHEMBL375076 0.71 CARM1 (0.56) BCHEACHEBACE1CARM1PRMT6
SCHEMBL2466378 0.70 CARM1 (0.68) BCHEACHEBACE1CARM1PRMT6
SCHEMBL375074 0.70 POLB (0.47) EPAS1ALDH1A1OPRL1POLBMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8623898-B2 Glycine transporter inhibiting substances TAISHO PHARMACEUTICAL CO., LTD. (JP) 2014-01-07 US disclosed
EP-2409976-A1 GLYCINE TRANSPORTER INHIBITOR Taisho Pharmaceutical Co., Ltd. (JP) 2012-01-25 EP disclosed
US-20120010414-A1 GLYCINE TRANSPORTER INHIBITING SUBSTANCES TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010414-A1 GLYCINE TRANSPORTER INHIBITING SUBSTANCES SLC18A2, SLC1A2, SLC6A1 BCHE 593/4885ACHE 467/4885BACE1 132/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.