SCHEMBL3757174

SCHEMBL3757174

COCCN(CCn1cc(-c2cc3nccc(Oc4ccc(N)cc4F)c3s2)cn1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.47
KDR P35968 12/20 0.47
MST1R Q04912 11/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2534756 0.91 MST1R (0.47) METKDRMST1R
SCHEMBL3568097 0.90 MET (0.51) METKDRMST1R
SCHEMBL2670833 0.89 MET (0.46) METKDRMST1R
SCHEMBL2670836 0.89 MET (0.46) METKDRMST1R
SCHEMBL10164514 0.84 MET (0.44) METKDRMST1R
SCHEMBL16187724 0.83 MET (0.52) METKDRMST1R
SCHEMBL2530838 0.83 MET (0.48) METKDRMST1R
SCHEMBL13166965 0.83 MET (0.46) METKDRMST1R
SCHEMBL2670642 0.82 MET (0.45) METKDRMST1R
SCHEMBL1674666 0.82 MST1R (0.43) METKDRMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183254-B1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY METHYLGENE INC (CA) 2017-06-21 EP disclosed
EP-2183254-A1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY MethylGene Inc. (CA) 2010-05-12 EP disclosed
WO-2009026717-A1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY METHYLGENE INC. (CA) 2009-03-05 WO disclosed