SCHEMBL3759645

SCHEMBL3759645

COC(=O)c1cc(Cc2ccccc2)c(C(C)C)n1Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.55
THRB P10828 3/20 0.55
KMT2A Q03164 2/20 0.45
GAA P10253 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
AR P10275 1/20 0.43
ALDH1A1 P00352 3/20 0.43
TSHR P16473 2/20 0.43
PKM P14618 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
TP53 P04637 3/20 0.42
POLB P06746 1/20 0.42
ATM Q13315 1/20 0.42
S1PR3 Q99500 1/20 0.42
HSP90AA1 P07900 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3757153 0.79 MAPK8 (0.47) MAPTTHRBKMT2AGAAL3MBTL1
SCHEMBL1884213 0.78 MAPT (0.46) MAPTTHRBKMT2AGAAL3MBTL1
SCHEMBL1877442 0.75 MAPT (0.49) MAPTTHRBKMT2AGAAL3MBTL1
SCHEMBL7884326 0.75 KMT2A (0.72) MAPTTHRBKMT2A
SCHEMBL1882299 0.74 TSHR (0.55) MAPTTHRBKMT2AGAAL3MBTL1
SCHEMBL1880517 0.73 MAPT (0.47) MAPTTHRBKMT2AGAAL3MBTL1
SCHEMBL2684278 0.73 MAPT (0.53) MAPTTHRBKMT2AGAAL3MBTL1
SCHEMBL1880402 0.72 MAPT (0.46) MAPTTHRBKMT2AGAAL3MBTL1
SCHEMBL1875614 0.70 GAA (0.60) MAPTTHRBKMT2AGAAL3MBTL1
SCHEMBL336671 0.70 MAPT (0.73) MAPTTHRBKMT2AGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185506-A1 PYRROLE COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST OR ANTAGONIST BIOLOGICAL ACTIVITY Allergan, Inc. (US) 2010-05-19 EP disclosed
WO-2009026407-A1 PYRROLE COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST OR ANTAGONIST BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2009-02-26 WO disclosed