SCHEMBL3757153

SCHEMBL3757153

COC(=O)c1c(Cc2ccccc2)cc(C(C)C)n1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 7/20 0.47
MAPT P10636 2/20 0.47
THRB P10828 1/20 0.47
AR P10275 1/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 2/20 0.44
PKM P14618 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
HSP90AA1 P07900 1/20 0.42
KDM4E B2RXH2 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPK9 P45984 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3756783 0.87 NOTUM (0.44) ALDH1A1GAAPKMSMN1; SMN2L3MBTL1
SCHEMBL1880517 0.80 MAPT (0.47) MAPK8MAPTTHRBARALDH1A1
SCHEMBL3759645 0.79 MAPT (0.55) MAPTTHRBARALDH1A1GAA
SCHEMBL1877442 0.76 MAPT (0.49) MAPK8MAPTTHRBARALDH1A1
SCHEMBL1875614 0.76 GAA (0.60) MAPK8MAPTTHRBARALDH1A1
SCHEMBL1890367 0.74 GAA (0.48) MAPK8MAPTTHRBARALDH1A1
SCHEMBL1884213 0.73 MAPT (0.46) MAPK8MAPTTHRBARALDH1A1
SCHEMBL182807 0.73 MAPK8 (0.57) MAPK8MAPTTHRBARALDH1A1
SCHEMBL1887533 0.71 MAPK8 (0.50) MAPK8MAPTTHRBARALDH1A1
SCHEMBL1884680 0.70 NOTUM (0.51) ALDH1A1GAAKDM4EKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185506-A1 PYRROLE COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST OR ANTAGONIST BIOLOGICAL ACTIVITY Allergan, Inc. (US) 2010-05-19 EP disclosed
WO-2009026407-A1 PYRROLE COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST OR ANTAGONIST BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2009-02-26 WO disclosed