SCHEMBL3760955

SCHEMBL3760955

Cc1ccc(-c2cnc3[nH]cc(-c4ccc(C(=O)O)c(F)c4)c3c2)cc1C

nearest known ligand 0.78

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AXL P30530 7/20 0.78
CAMKK2 Q96RR4 6/20 0.71
PIK3CG P48736 3/20 0.61
SGK1 O00141 5/20 0.60
DYRK1A Q13627 3/20 0.56
AURKA O14965 1/20 0.53
CAMKK1 Q8N5S9 1/20 0.53
SGK3 Q96BR1 1/20 0.53
SGK2 Q9HBY8 1/20 0.53
NTRK1 P04629 1/20 0.50
CLK1 P49759 1/20 0.50
CLK2 P49760 1/20 0.50
DYRK2 Q92630 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
DYRK1B Q9Y463 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3770773 0.91 CAMKK2 (0.85) AXLCAMKK2PIK3CGSGK1DYRK1A
SCHEMBL3763876 0.85 AXL (0.72) AXLCAMKK2PIK3CGSGK1DYRK1A
SCHEMBL3763368 0.85 AXL (0.82) AXLCAMKK2PIK3CGSGK1DYRK1A
SCHEMBL3771696 0.84 AXL (0.74) AXLCAMKK2PIK3CGSGK1DYRK1A
SCHEMBL3769565 0.84 AXL (0.76) AXLCAMKK2SGK1NTRK1
SCHEMBL3763779 0.84 AXL (0.70) AXLCAMKK2SGK1DYRK1A
SCHEMBL3767383 0.83 CAMKK2 (1.00) AXLCAMKK2SGK1AURKACAMKK1
SCHEMBL3774334 0.83 AXL (0.74) AXLCAMKK2PIK3CGSGK1AURKA
SCHEMBL3763777 0.83 AXL (0.76) AXLCAMKK2PIK3CGSGK1DYRK1A
SCHEMBL3766333 0.83 AXL (0.74) AXLCAMKK2PIK3CGSGK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120238588-A1 1H-Pyrrolo[2,3-B]Pyridines GlaxoSmithKline, LLC 2012-09-20 US claimed
WO-2010049173-A1 USE OF INHIBITORS OF HOST KINASES FOR THE TREATMENT OF INFECTIOUS DISEASES CENIX BIOSCIENCE GMBH (DE) 2010-05-06 WO claimed
US-20090233955-A1 1H-Pyrrolo[2,3-B]Pyridnes GLAXOSMITHKLINE LLC 2009-09-17 US claimed
EP-1828180-A1 1H-PYRROLO[2,3-BETA]PYRIDINES SMITHKLINE BEECHAM CORPORATION (US) 2007-09-05 EP claimed
WO-2006063167-A1 1H-PYRROLO[2,3-B]PYRIDINES SMITHKLINE BEECHAM CORPORATION (US) 2006-06-15 WO claimed
WO-2021006707-A1 USE OF SGK1 INHIBITOR AS THERAPEUTIC AGENT FOR INFLAMMATORY NEUROLOGICAL DISEASES 한양대학교 산학협력단 2021-01-14 WO disclosed
US-20120238588-A1 1H-Pyrrolo[2,3-B]Pyridines GlaxoSmithKline, LLC 2012-09-20 US disclosed
WO-2010049173-A1 USE OF INHIBITORS OF HOST KINASES FOR THE TREATMENT OF INFECTIOUS DISEASES CENIX BIOSCIENCE GMBH (DE) 2010-05-06 WO disclosed
US-20090233955-A1 1H-Pyrrolo[2,3-B]Pyridnes GLAXOSMITHKLINE LLC 2009-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233955-A1 1H-Pyrrolo[2,3-B]Pyridnes SGK1, SGK2, SGK3 AXL 1542/4885CAMKK2 157/4885PIK3CG 377/4885
US-20120238588-A1 1H-Pyrrolo[2,3-B]Pyridines SGK1, SGK2, SGK3 AXL 1432/4885CAMKK2 125/4885PIK3CG 393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.