SCHEMBL3767702

SCHEMBL3767702

Fc1cc(CN2CCC2)ccc1-c1cc2cc(Cc3ccccn3)ccc2o1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 12/20 0.56
S1PR3 Q99500 6/20 0.56
KCNH2 Q12809 1/20 0.56
MAOB P27338 2/20 0.44
CXCR4 P61073 1/20 0.40
CHKA P35790 3/20 0.39
MAOA P21397 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
PRKCQ Q04759 1/20 0.36
PRKCD Q05655 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1602472 0.86 S1PR1 (0.79) S1PR1S1PR3KCNH2
SCHEMBL3696705 0.82 S1PR1 (0.51) S1PR1S1PR3KCNH2MAOBCHKA
SCHEMBL1602805 0.81 S1PR1 (0.63) S1PR1S1PR3KCNH2
SCHEMBL3706283 0.80 S1PR1 (0.60) S1PR1S1PR3KCNH2MAOBCHKA
SCHEMBL3772064 0.77 S1PR1 (0.53) S1PR1S1PR3KCNH2MAOBCHKA
SCHEMBL3706281 0.75 S1PR1 (0.52) S1PR1S1PR3KCNH2MAOBCHKA
SCHEMBL1602487 0.75 S1PR1 (0.80) S1PR1S1PR3KCNH2
SCHEMBL1602394 0.73 S1PR1 (0.85) S1PR1S1PR3KCNH2MAOB
SCHEMBL1601448 0.73 S1PR1 (0.85) S1PR1S1PR3KCNH2MAOB
SCHEMBL4442277 0.72 S1PR1 (0.55) S1PR1S1PR3KCNH2MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2010522162-A 2010-07-01 JP claimed
EP-2121648-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX Pharmaceuticals, Inc. (US) 2009-11-25 EP claimed
WO-2007109334-A2 SIP RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-09-27 WO claimed