SCHEMBL3706283

SCHEMBL3706283

Fc1cc(CN2CCC2)ccc1-c1cc2cc(CCCc3ccccc3)ccc2o1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 11/20 0.60
S1PR3 Q99500 5/20 0.60
KCNH2 Q12809 1/20 0.60
MAOB P27338 1/20 0.46
CHKA P35790 2/20 0.42
DRD2 P14416 3/20 0.41
HTR2B P41595 2/20 0.41
DRD4 P21917 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4440616 0.85 S1PR1 (0.82) S1PR1S1PR3KCNH2
SCHEMBL3772064 0.82 S1PR1 (0.53) S1PR1S1PR3KCNH2MAOBCHKA
SCHEMBL4443009 0.81 S1PR1 (0.85) S1PR1S1PR3KCNH2
SCHEMBL4446551 0.81 S1PR1 (0.69) S1PR1S1PR3KCNH2MAOB
SCHEMBL3706281 0.80 S1PR1 (0.52) S1PR1S1PR3KCNH2MAOBCHKA
SCHEMBL3767702 0.80 S1PR1 (0.56) S1PR1S1PR3KCNH2MAOBCHKA
SCHEMBL12730038 0.79 S1PR1 (0.69) S1PR1S1PR3CHKAHTR2BKMT2A
SCHEMBL4449544 0.77 S1PR1 (0.71) S1PR1S1PR3KCNH2MAOB
SCHEMBL1601448 0.76 S1PR1 (0.85) S1PR1S1PR3KCNH2MAOB
SCHEMBL1602394 0.76 S1PR1 (0.85) S1PR1S1PR3KCNH2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2010522162-A 2010-07-01 JP claimed
EP-2121648-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX Pharmaceuticals, Inc. (US) 2009-11-25 EP claimed
WO-2007109334-A2 SIP RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-09-27 WO claimed