SCHEMBL3767950

SCHEMBL3767950

O=C(COc1ccc2ccccc2c1)N1CCN(CC(=O)N2CCN(C3CCC3)CC2)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.70
NPC1 O15118 1/20 0.63
HPGD P15428 1/20 0.63
RAB9A P51151 1/20 0.63
KDM4E B2RXH2 3/20 0.60
GPR183 P32249 1/20 0.57
LMNA P02545 2/20 0.54
GAA P10253 2/20 0.54
MAPT P10636 2/20 0.54
ALOX15 P16050 1/20 0.54
ALDH1A1 P00352 6/20 0.54
ACHE P22303 3/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
POLB P06746 2/20 0.53
GLA P06280 1/20 0.53
USP2 O75604 1/20 0.53
TP53 P04637 1/20 0.53
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4384365 0.91 SMN1; SMN2 (0.74) SMN1; SMN2NPC1HPGDRAB9AKDM4E
SCHEMBL4381637 0.90 SMN1; SMN2 (0.73) SMN1; SMN2NPC1HPGDRAB9AKDM4E
SCHEMBL3774181 0.88 KDM4E (0.78) SMN1; SMN2KDM4ELMNAGAAMAPT
SCHEMBL3769014 0.85 KDM4E (0.55) SMN1; SMN2NPC1RAB9AKDM4EACHE
SCHEMBL2831262 0.84 NPC1 (0.76) SMN1; SMN2NPC1HPGDRAB9AKDM4E
SCHEMBL3779346 0.84 NPSR1 (0.72) SMN1; SMN2NPC1RAB9AKDM4ELMNA
SCHEMBL3767792 0.84 KDM4E (0.59) SMN1; SMN2KDM4EMAPTACHEMEN1
SCHEMBL3776429 0.84 GAA (0.61) SMN1; SMN2KDM4ELMNAGAAALDH1A1
SCHEMBL3774220 0.84 KDM4E (0.61) SMN1; SMN2HPGDRAB9AKDM4EGPR183
SCHEMBL3767766 0.84 ACHE (0.68) SMN1; SMN2KDM4EALOX15ALDH1A1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851474-B2 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION (US) 2010-12-14 US disclosed
US-7851474-B2 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION (US) 2010-12-14 US disclosed
US-7851474-B2 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION (US) 2010-12-14 US disclosed
US-20070049571-A1 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION 2007-03-01 US disclosed
US-20070049571-A1 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION 2007-03-01 US disclosed
US-20070049571-A1 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION 2007-03-01 US disclosed
WO-2007016496-A2 DIPIPERAZINYL KETONES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2007-02-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070049571-A1 Dipiperazinyl ketones and related analogues HRH4, HRH3, HRH1 SMN1; SMN2 4282/4885NPC1 3462/4885HPGD 377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.