SCHEMBL3772890

SCHEMBL3772890

CC(C)(C)OC(=O)N1CCN2C(=O)COCC2C1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.44
USP2 O75604 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
RECQL P46063 1/20 0.39
SMARCA2 P51531 1/20 0.38
SMARCA4 P51532 1/20 0.38
PBRM1 Q86U86 1/20 0.38
PIK3CD O00329 2/20 0.38
GPR119 Q8TDV5 1/20 0.37
TP53 P04637 1/20 0.37
FPR2 P25090 2/20 0.37
PIK3R1 P27986 3/20 0.37
PIK3CA P42336 3/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL994944 1.00 USP30 (0.44) USP30USP2SMN1; SMN2RECQLSMARCA2
SCHEMBL9978161 1.00 USP30 (0.44) USP30USP2SMN1; SMN2RECQLSMARCA2
SCHEMBL2943987 0.81 USP30 (0.43) USP30USP2SMN1; SMN2RECQLGPR119
SCHEMBL2954128 0.81 USP30 (0.43) USP30USP2SMN1; SMN2RECQLGPR119
SCHEMBL780002 0.81 USP30 (0.43) USP30USP2SMN1; SMN2RECQLGPR119
SCHEMBL23422324 0.80 USP30 (0.47) USP30USP2SMN1; SMN2SMARCA2SMARCA4
SCHEMBL14815454 0.80 USP30 (0.47) USP30USP2SMN1; SMN2SMARCA2SMARCA4
SCHEMBL31027198 0.80 USP30 (0.47) USP30USP2SMN1; SMN2SMARCA2SMARCA4
SCHEMBL1441275 0.79 USP2 (0.48) USP30USP2SMN1; SMN2RECQLPIK3CD
SCHEMBL3774805 0.79 PIK3CD (0.39) SMN1; SMN2PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940845-B1 NOVEL AZETIDINE COMPOUNDS USEFUL IN THE TREATMENT OF FUNCTIONAL GASTROINTESTINAL DISORDERS, IBS AND FUNCTIONAL DYSPEPSIA ALBIREO AB (SE) 2013-06-12 EP claimed
US-20250026758-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS INC (US) 2025-01-23 US disclosed
CN-119112895-A Muscarinic acetylcholine M1 receptor antagonists 康蒂内乌姆医疗公司 2024-12-13 CN disclosed
CN-112638381-B Muscarinic acetylcholine M1 receptor antagonists 康蒂内乌姆医疗公司 2024-08-30 CN disclosed
US-12054487-B2 Muscarinic acetylcholine M1 receptor antagonists CONTINEUM THERAPEUTICS, INC. (US) 2024-08-06 US disclosed
WO-2023067355-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LIMITED (GB) 2023-04-27 WO disclosed
EP-3846806-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS Pipeline Therapeutics, Inc. (US) 2021-07-14 EP disclosed
US-20210155629-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS, INC. 2021-05-27 US disclosed
US-20210155629-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS, INC. 2021-05-27 US disclosed
CN-112638381-A Muscarinic acetylcholine M1 receptor antagonists 帕珀莱恩医疗公司 2021-04-09 CN disclosed
EP-1940845-B1 NOVEL AZETIDINE COMPOUNDS USEFUL IN THE TREATMENT OF FUNCTIONAL GASTROINTESTINAL DISORDERS, IBS AND FUNCTIONAL DYSPEPSIA ALBIREO AB (SE) 2013-06-12 EP disclosed
US-8288370-B2 Substituted azetidine compounds of formula (I) useful in the treatment of functional gastrointestinal disorders, IBS, and functional dyspepsia ALBIREO AB (SE) 2012-10-16 US disclosed
US-20100311713-A1 Novel Azetidine Compounds Useful in the Treatment of Functional Gastrointestinal Disorders, Ibs and Functional Dyspepsia ASTRAZENECA AB (SE) 2010-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210155629-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CHRM1, CHRM2, CHRM5 USP30 2387/4885USP2 2496/4885SMN1; SMN2 1028/4885
US-20100311713-A1 Novel Azetidine Compounds Useful in the Treatment of Functional Gastrointestinal Disorders, Ibs and Functional Dyspepsia NISCH, BDKRB2, VIP USP30 1738/4885USP2 1988/4885SMN1; SMN2 3177/4885
US-12054487-B2 Muscarinic acetylcholine M1 receptor antagonists CHRM1, CHRM2, CHRM3 USP30 2186/4885USP2 2885/4885SMN1; SMN2 1266/4885
US-20250026758-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CHRM1, CHRM2, CHRM5 USP30 2387/4885USP2 2496/4885SMN1; SMN2 1028/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.