SCHEMBL3779802

SCHEMBL3779802

COC(=O)C1=C(C(=O)OC)C(=O)CC=N1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.33
FGFR1 P11362 3/20 0.32
FGFR2 P21802 3/20 0.32
FGFR4 P22455 3/20 0.32
FGFR3 P22607 3/20 0.32
SRC P12931 2/20 0.32
HPGD P15428 2/20 0.31
LMNA P02545 1/20 0.31
KDM4E B2RXH2 2/20 0.31
MAPK1 P28482 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP3A4 P08684 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6885396 0.78 MAPT (0.38) NPSR1HPGDLMNACYP3A4ALDH1A1
SCHEMBL8557965 0.76 NPSR1 (0.37) NPSR1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL31333069 0.67 CHRM3 (0.40) NPSR1LMNAKDM4EALDH1A1TSHR
SCHEMBL19297097 0.62 NPSR1 (0.34) NPSR1KDM4EMAPK1ALDH1A1TSHR
SCHEMBL9242569 0.61 NPSR1 (0.46) NPSR1FGFR1FGFR2FGFR4FGFR3
SCHEMBL7311210 0.61 NPSR1 (0.33) NPSR1FGFR1FGFR2FGFR4FGFR3
SCHEMBL9292998 0.60 NPSR1 (0.41) NPSR1LMNAKDM4EMAPK1L3MBTL1
SCHEMBL5798986 0.58
SCHEMBL22570267 0.58
SCHEMBL5344290 0.58 CHRM3 (0.39) NPSR1HPGDLMNAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2187893-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2010-05-26 EP disclosed
WO-2009111676-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS ANACOR PHARMACEUTICALS, INC (US) 2009-09-11 WO disclosed