SCHEMBL3782097

SCHEMBL3782097

OCC#Cc1ccc2nc(-c3ccco3)nc(N[C@H]3CC[C@H](O)CC3)c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.47
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
TDP1 Q9NUW8 3/20 0.40
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
GLA P06280 2/20 0.40
RECQL P46063 2/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
ADORA1 P30542 6/20 0.39
ADORA2A P29274 4/20 0.39
ADORA3 P0DMS8 3/20 0.39
ADORA2B P29275 1/20 0.39
PDE5A O76074 2/20 0.38
CYP1A2 P05177 5/20 0.37
CYP3A4 P08684 5/20 0.37
CLK4 Q9HAZ1 5/20 0.37
USP2 O75604 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3782101 1.00 GBA1 (0.47) GBA1MEN1KMT2ATDP1ALDH1A1
SCHEMBL3806943 0.90 GBA1 (0.52) GBA1MEN1KMT2ATDP1ALDH1A1
SCHEMBL3806946 0.90 GBA1 (0.52) GBA1MEN1KMT2ATDP1ALDH1A1
SCHEMBL3706548 0.81 PDE5A (0.47) GBA1ADORA1ADORA2AADORA3ADORA2B
SCHEMBL3708230 0.81 PDE5A (0.61) GBA1MEN1KMT2AALDH1A1KDM4E
SCHEMBL3706663 0.80 CCNE2 (0.48) GBA1MEN1KMT2AALDH1A1ADORA1
SCHEMBL30772425 0.80 PDE5A (0.41) GBA1MEN1KMT2ATDP1ALDH1A1
SCHEMBL2803755 0.80 PDE5A (0.41) GBA1MEN1KMT2ATDP1ALDH1A1
SCHEMBL13283709 0.75 GBA1 (0.46) GBA1MEN1KMT2ATDP1ALDH1A1
SCHEMBL3809901 0.69 PDE5A (0.49) GBA1MEN1KMT2ATDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010081881-A1 AURORA KINASE INHIBITORS COMPOUNDS. UNIVERSITÄT LEIPZIG (DE) 2010-07-22 WO claimed
WO-2010081881-A1 AURORA KINASE INHIBITORS COMPOUNDS. UNIVERSITÄT LEIPZIG (DE) 2010-07-22 WO disclosed