SCHEMBL3788362

SCHEMBL3788362

O=C(O)Cn1nc2ccc(C(=O)NCc3ccccc3OC(F)(F)F)cn2c1=O

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.49
PPARG P37231 2/20 0.49
ROCK2 O75116 2/20 0.47
ROCK1 Q13464 1/20 0.47
RIPK1 Q13546 7/20 0.47
GPR139 Q6DWJ6 2/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HSD17B13 Q7Z5P4 3/20 0.43
NTRK1 P04629 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3811009 0.93 EPHX2 (0.48) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL3796727 0.91 EPHX2 (0.52) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL3790889 0.90 PPARG (0.52) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL13258052 0.90 EPHX2 (0.49) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL3786599 0.90 EPHX2 (0.48) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL3786760 0.90 EPHX2 (0.48) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL3788636 0.89 EPHX2 (0.48) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL3788935 0.88 EPHX2 (0.47) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL3791605 0.88 EPHX2 (0.49) EPHX2PPARGROCK2ROCK1RIPK1
SCHEMBL3794154 0.87 EPHX2 (0.52) EPHX2PPARGROCK2ROCK1RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed