SCHEMBL3789154

SCHEMBL3789154

Cc1nc2ccc(-c3ccc4c(c3)CN(C(=O)N3CCCCC3c3ccc(OC(F)(F)F)cc3)CCO4)cc2[nH]1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 15/20 0.57
SCD5 Q86SK9 1/20 0.42
HCRTR1 O43613 2/20 0.40
HCRTR2 O43614 2/20 0.40
CREBBP Q92793 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3799784 0.92 PIK3CA (0.54) PIK3CASCD5HCRTR1HCRTR2CREBBP
SCHEMBL2725828 0.91 PIK3CA (0.59) PIK3CAHCRTR1HCRTR2CREBBP
SCHEMBL2733019 0.90 PIK3CA (0.57) PIK3CASCD5CREBBP
SCHEMBL3791617 0.90 PIK3CA (0.56) PIK3CACREBBP
SCHEMBL3798622 0.89 PIK3CA (0.55) PIK3CACREBBP
SCHEMBL7881809 0.88 PIK3CA (0.56) PIK3CACREBBP
SCHEMBL6126363 0.88 PIK3CA (0.56) PIK3CACREBBP
SCHEMBL2724235 0.88 PIK3CA (0.56) PIK3CACREBBP
SCHEMBL2727770 0.88 PIK3CA (0.59) PIK3CACREBBP
SCHEMBL7880624 0.88 PIK3CA (0.56) PIK3CACREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010138490-A1 BENZOXAZEPINES AS INHIBITORS OF MTOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2010-12-02 WO disclosed