SCHEMBL3789170

SCHEMBL3789170

Cc1noc(C(Cc2c[nH]c3ccccc23)NC(=O)O)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 4/20 0.50
MAPT P10636 4/20 0.50
KDM4E B2RXH2 2/20 0.50
POLB P06746 2/20 0.50
APAF1 O14727 1/20 0.50
RECQL P46063 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
ITGB2 P05107 1/20 0.48
ICAM1 P05362 1/20 0.48
ITGAL P20701 1/20 0.48
ALOX15 P16050 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ACE P12821 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
MPO P05164 1/20 0.47
TSHR P16473 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4115544 0.87 P4HB (0.64) SRCMAPTPOLBSMN1; SMN2ACE
SCHEMBL21062749 0.85 SRC (0.64) SRCSMN1; SMN2MEN1KMT2A
SCHEMBL21062751 0.85 SRC (0.64) SRCSMN1; SMN2MEN1KMT2A
SCHEMBL6723448 0.83 POLB (0.53) MAPTKDM4EPOLBAPAF1RECQL
SCHEMBL21062784 0.82 SRC (0.62) SRCSMN1; SMN2
SCHEMBL21062785 0.82 SRC (0.62) SRCSMN1; SMN2
SCHEMBL20510013 0.81 P4HB (0.57) MAPTKDM4EPOLBAPAF1RECQL
SCHEMBL20510012 0.81 P4HB (0.57) MAPTKDM4EPOLBAPAF1RECQL
SCHEMBL28910646 0.79 SRC (0.47) SRC
SCHEMBL28910647 0.79 SRC (0.47) SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260022-B1 SUBSTITUTED CYCLOHEXYLDIAMINES GRUENENTHAL GMBH (DE) 2017-01-04 EP disclosed
EP-2260022-A1 SUBSTITUTED CYCLOHEXYLDIAMINES Grünenthal GmbH (DE) 2010-12-15 EP disclosed
WO-2009118174-A1 SUBSTITUTED CYCLOHEXYLDIAMINES Grünenthal GmbH (DE) 2009-10-01 WO disclosed