Meglitinide

Meglitinide

SCHEMBL37926

COc1ccc(Cl)cc1C(=O)NCCc1ccc(C(=O)O)cc1

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DNMT3A Q9Y6K1 1/20 0.78
HDAC1 Q13547 2/20 0.72
HDAC6 Q9UBN7 2/20 0.72
NLRP3 Q96P20 3/20 0.71
GAA P10253 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Meglitinide SCHEMBL29829482 1.00 DNMT3A (0.78) DNMT3AHDAC1HDAC6NLRP3GAA
SCHEMBL11354611 0.91 DNMT3A (0.75) DNMT3AHDAC1HDAC6NLRP3GAA
SCHEMBL11360335 0.91 DNMT3A (0.78) DNMT3AHDAC1HDAC6NLRP3GAA
SCHEMBL11479096 0.90 HDAC1 (0.71) DNMT3AHDAC1HDAC6NLRP3
SCHEMBL1153776 0.90 DNMT3A (0.67) DNMT3AHDAC1HDAC6NLRP3
SCHEMBL3784241 0.89 DNMT3A (0.80) DNMT3AHDAC1HDAC6NLRP3
SCHEMBL8261934 0.89 DNMT3A (0.84) DNMT3AHDAC1HDAC6NLRP3
SCHEMBL1154792 0.88 DNMT3A (0.62) DNMT3AHDAC1HDAC6NLRP3GAA
SCHEMBL30381560 0.88 HDAC1 (0.79) DNMT3AHDAC1HDAC6NLRP3
SCHEMBL11481071 0.88 HDAC1 (0.79) DNMT3AHDAC1HDAC6NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12491 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260115210-A1 METHOD FOR TREATING SUBJECTS SUFFERING FROM CENTRAL NERVOUS SYSTEM CONTUSIONS REMEDY PHARMACEUTICALS, INC. (US) 2026-04-30 US claimed
EP-3634453-B1 PLANT EXTRACTS WITH ANTI-DIABETIC AND OTHER USEFUL ACTIVITIES HOUSEY PHARMACEUTICAL RES LABORATORIES L L C (US) 2026-04-29 EP claimed
US-12611401-B2 Combinations comprising benzodioxol as GLP-1R agonists for use in the treatment of NASH/NAFLD and related diseases PFIZER INC. (US) 2026-04-28 US claimed
US-12611416-B2 Methods of treating ischemic stroke at risk for cerebral or cerebellar edema REMEDY PHARMACEUTICALS, INC. (US) 2026-04-28 US claimed
US-12599564-B2 Antidiabetic pharmaceutical compositions Elite Pharmaceutical Solution Inc. (US) 2026-04-14 US claimed
US-20260069550-A1 TRANSDERMAL DELIVERY OF ANTIDIABETIC AGENTS RITTENHOUSE CHRISTINE (US) 2026-03-12 US claimed
EP-4705280-A1 DIARYL UREA-BASED COMPOUNDS AND RELATED COMPOSITIONS AND METHODS OF USE IN THE TREATMENT OF DIABETES MELLITUS AND NEURODEGENERATIVE DISEASE Purdue Research Foundation (US) 2026-03-11 EP claimed
EP-4699609-A2 HETEROCYCLIC GLP-1 AGONISTS Gasherbrum Bio, Inc. (US) 2026-02-25 EP claimed
US-12527754-B2 Methods and compositions for preventing and treating metabolic syndrome induced by antipsychotic treatment and related diseases and conditions TUFTS MEDICAL CENTER, INC. (US) 2026-01-20 US claimed
US-20250381199-A1 PHARMACEUTICAL PREPARATION FOR IMPROVING ABSORPTION AND POSTPRANDIAL HYPOGLYCEMIC ACTION OF INSULIN LILLY CO ELI (US) 2025-12-18 US claimed
WO-2001055085-A1 PROPIONIC ACID DERIVATIVES AND THEIR USE IN THE TREATMENT OF DIABETES AND OBESITY NOVO NORDISK A/S (DK) 2001-08-02 WO claimed
WO-2001055086-A1 ALKYNYLSUBSTITUTED PROPIONIC ACID DERIVATIVES AND THEIR USE AGAINST DIABETES AND OBESITY NOVO NORDISK A/S (DK) 2001-08-02 WO claimed
WO-2001032158-A2 PHARMACEUTICAL COMPOSITION COMPRISING A COMBINATION OF METFORMIN AND ANOTHER ANTIDIABETIC AGENT BRISTOL-MYERS SQUIBB COMPANY (US) 2001-05-10 WO claimed
WO-2001027128-A1 C-ARYL GLUCOSIDE SGLT2 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-04-19 WO claimed
WO-2001027107-A2 HETEROCYCLIC SODIUM/PROTON EXCHANGE INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2001-04-19 WO claimed
EP-1088824-A2 Bicyclic pyrrolyl amides as glycogen phosphorylase inhibitors Pfizer Products Inc. (US) 2001-04-04 EP claimed
WO-2001021602-A1 OXA- AND THIAZOLE DERIVATIVES USEFUL AS ANTIDIABETIC AND ANTIOBESITY AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-03-29 WO claimed
WO-2000059506-A1 HETEROCYCLIC CONTAINING BIPHENYL aP2 INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB CO. (US) 2000-10-12 WO claimed
WO-2000015229-A1 METHOD FOR TREATING DIABETES EMPLOYING AN aP2 INHIBITOR AND COMBINATION BRISTOL-MYERS SQUIBB COMPANY (US) 2000-03-23 WO claimed
US-4221815-A HYPOGLYCEMIC AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1980-09-09 US claimed