SCHEMBL379265

SCHEMBL379265

COc1ccc(C(F)(F)F)cc1NC(=O)Nc1c(F)cccc1/C=C(\C)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 10/20 0.46
POLB P06746 1/20 0.43
MAPK14 Q16539 1/20 0.43
KDM4E B2RXH2 3/20 0.43
HPGD P15428 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
ATM Q13315 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
BRAF P15056 1/20 0.42
HTT P42858 1/20 0.41
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDR P35968 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16428166 1.00 RAF1 (0.46) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL379266 1.00 RAF1 (0.46) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL4534203 0.85 RAF1 (0.47) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL4534200 0.85 RAF1 (0.47) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL27145420 0.85 RAF1 (0.47) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL15229756 0.83 RAF1 (0.47) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL28799154 0.83 RAF1 (0.47) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL379165 0.83 RAF1 (0.47) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL30667504 0.83 RAF1 (0.47) RAF1POLBMAPK14KDM4EHPGD
SCHEMBL31686438 0.83 RAF1 (0.51) RAF1POLBMAPK14KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893587-B1 METHOD FOR PRODUCING DIHYDROQUINAZOLINES AICURIS GMBH & CO KG (DE) 2012-01-25 EP claimed
US-8084604-B2 Process for the preparation of dihydroquinazolines Aicuris GmbH & Co., KG (DE) 2011-12-27 US claimed
US-8084604-B2 Process for the preparation of dihydroquinazolines Aicuris GmbH & Co., KG (DE) 2011-12-27 US disclosed