SCHEMBL379502

SCHEMBL379502

NC(c1ccccn1)c1nccc2scc(Br)c12

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KDR P35968 2/20 0.32
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL380700 0.83 KDR (0.44) KDRAURKAAURKB
SCHEMBL2368686 0.80 EGFR (0.37) SLC6A2SLC6A4SLC6A3KDRAURKB
SCHEMBL379684 0.79 AURKA (0.33) KDRAURKAAURKB
SCHEMBL379851 0.78 MAPT (0.38) KDRAURKAAURKB
SCHEMBL1131039 0.69 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL6775513 0.67 SLC6A2 (0.52) SLC6A2SLC6A4SLC6A3
Methane SCHEMBL28543758 0.67 SLC6A2 (0.52) SLC6A2SLC6A4SLC6A3
SCHEMBL868356 0.67 KDR (0.57) KDRAURKAAURKB
SCHEMBL29503401 0.67 KDR (0.57) KDRAURKAAURKB
SCHEMBL18341971 0.66 KDR (0.40) KDRAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9216992-B2 Thieno[3,2-c]pyridine potassium channel inhibitors XENTION LIMITED (GB) 2015-12-22 US disclosed
EP-1968982-B1 THIENO (3,2-C) PYRIDINE COMPOUNDS XENTION LTD (GB) 2012-01-25 EP disclosed
EP-1968982-A2 THIENO (3,2-C) PYRIDINE COMPOUNDS Xention Discovery Ltd. (GB) 2008-09-17 EP disclosed
US-20070161672-A1 Compounds XENTION LIMITED 2007-07-12 US disclosed
WO-2007066127-A2 THIENO ( 3 , 2-C) PYRIDINE COMPOUNDS XENTION LIMITED (GB) 2007-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070161672-A1 Compounds KCNJ2, KCNT1, KCNT2 SLC6A2 2905/4885SLC6A4 3095/4885SLC6A3 3100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.