SCHEMBL379647

SCHEMBL379647

NC(=O)CCCCNCCc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.65
ADRB2 P07550 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CHRM1 P11229 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
DRD1 P21728 1/20 0.54
SLC6A2 P23975 1/20 0.54
SLC6A4 P31645 1/20 0.54
ADRA1A P35348 1/20 0.54
PTGS2 P35354 1/20 0.54
HRH1 P35367 1/20 0.54
DRD3 P35462 1/20 0.54
OPRK1 P41145 1/20 0.54
SLC6A3 Q01959 1/20 0.54
PDE4D Q08499 1/20 0.54
KCNH2 Q12809 1/20 0.54
HRH3 Q9Y5N1 1/20 0.54
HDAC1 Q13547 1/20 0.53
HDAC2 Q92769 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3824789 0.89 SIGMAR1 (0.55) SIGMAR1OPRK1HDAC1HDAC2
SCHEMBL10766680 0.86 SIGMAR1 (0.66) SIGMAR1
SCHEMBL13584782 0.83 MAPT (0.61) ADRA1ASLC6A3HDAC1HDAC2
SCHEMBL10453660 0.83 SIGMAR1 (0.91) SIGMAR1ADRB2ADORA3CHRM1ADRA2B
SCHEMBL2872694 0.82 SIGMAR1 (0.66) SIGMAR1ADRA1ASLC6A3HDAC1HDAC2
SCHEMBL11232716 0.82 MAPT (0.57) SIGMAR1HDAC1HDAC2
SCHEMBL19438542 0.82 SIGMAR1 (0.59) SIGMAR1
SCHEMBL10436247 0.81 HDAC3 (0.74) HDAC1HDAC2
SCHEMBL1285919 0.81 MAPT (0.70) ADRA1ASLC6A3HDAC1HDAC2
SCHEMBL20689719 0.81 SIGMAR1 (0.91) SIGMAR1ADRB2ADORA3CHRM1ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408450-A1 A NOVEL ALPHA-(N-SULFONAMIDO)ACETAMIDE COMPOUND AS AN INHIBITOR OF BETA AMYLOID PEPTIDE PRODUCTION Bristol-Myers Squibb Company (US) 2012-01-25 EP disclosed
WO-2010107435-A1 A NOVEL ALPHA-(N-SULFONAMIDO)ACETAMIDE COMPOUND AS AN INHIBITOR OF BETA AMYLOID PEPTIDE PRODUCTION BRISTOL-MYERS SQUIBB COMPANY (US) 2010-09-23 WO disclosed