SCHEMBL3797322

SCHEMBL3797322

Cc1c(C(=O)O)cccc1-n1c(C)nc2ccc(C(F)(F)F)cc21

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
POLB P06746 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
SORT1 Q99523 4/20 0.44
DHODH Q02127 2/20 0.44
NOTUM Q6P988 1/20 0.43
TP53 P04637 1/20 0.41
TAS2R14 Q9NYV8 1/20 0.40
BMI1 P35226 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
GRIK1 P39086 1/20 0.37
MYC P01106 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3792099 0.91 HSD17B10 (0.44) ALDH1A1L3MBTL1POLBTDP1SORT1
SCHEMBL1708022 0.88 ALDH1A1 (0.48) ALDH1A1POLBSORT1DHODHTP53
SCHEMBL1708275 0.81 BMI1 (0.37) ALDH1A1L3MBTL1DHODHBMI1
SCHEMBL1708107 0.79 TSHR (0.46) ALDH1A1POLBTP53MRGPRX4MYC
SCHEMBL1708108 0.72 POLB (0.53) ALDH1A1L3MBTL1POLBTP53MYC
SCHEMBL28464972 0.71 TSHR (0.67) ALDH1A1L3MBTL1POLBTP53
SCHEMBL1356522 0.69 HSD17B10 (0.64) ALDH1A1L3MBTL1POLBTDP1NOTUM
SCHEMBL27715912 0.68 TRPV1 (0.46) ALDH1A1SORT1NOTUMTAS2R14MRGPRX4
SCHEMBL12135484 0.67 KMT2A (0.50) ALDH1A1L3MBTL1POLBTDP1DHODH
SCHEMBL15727582 0.67 KDM4E (0.50) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed