SCHEMBL3799358

SCHEMBL3799358

C#CCN(C)Cc1ccc(NC(=O)OC23CC4CC(C)(CC(C)(C4)C2)C3)c2ncccc12

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.51
BCHE P06276 3/20 0.51
MAOA P21397 8/20 0.48
MAOB P27338 8/20 0.48
BACE1 P56817 1/20 0.48
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
KDM4E B2RXH2 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CTSB P07858 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL608500 0.79 ACHE (0.63) ACHEBCHEMAOAMAOBBACE1
SCHEMBL609576 0.77 ACHE (0.61) ACHEBCHEMAOAMAOBBACE1
SCHEMBL611410 0.74 ACHE (0.53) ACHEBCHEMAOAMAOBBACE1
SCHEMBL611971 0.74 ACHE (0.53) ACHEBCHEMAOAMAOBBACE1
SCHEMBL608172 0.71 ACHE (0.68) ACHEBCHEMAOAMAOBBACE1
SCHEMBL608563 0.70 ACHE (0.71) ACHEBCHEMAOAMAOBBACE1
SCHEMBL608751 0.69 ACHE (0.81) ACHEBCHEMAOAMAOBBACE1
SCHEMBL608520 0.69 ACHE (1.00) ACHEBCHEMAOAMAOBBACE1
SCHEMBL608665 0.68 ACHE (0.75) ACHEBCHEMAOAMAOBBACE1
SCHEMBL608173 0.68 ACHE (0.68) ACHEBCHEMAOAMAOBBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010086860-A2 NEUROPROTECTIVE MULTIFUNCTIONAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2010-08-05 WO disclosed