SCHEMBL3799564

SCHEMBL3799564

COc1c(C)cnc(CS(=O)(=O)O)c1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGXT P21549 1/20 0.57
CYP2C9 P11712 2/20 0.53
KMT2A Q03164 4/20 0.44
WDR5 P61964 3/20 0.44
PDE10A Q9Y233 1/20 0.42
ATP4A P20648 3/20 0.42
ATP4B P51164 3/20 0.42
DDAH1 O94760 2/20 0.42
BRS3 P32247 2/20 0.42
ENGASE Q8NFI3 2/20 0.42
ATP1A1 P05023 2/20 0.42
ATP1B1 P05026 2/20 0.42
ATP1A3 P13637 2/20 0.42
ATP1B2 P14415 2/20 0.42
ATP1A2 P50993 2/20 0.42
ATP1B3 P54709 2/20 0.42
FXYD2 P54710 2/20 0.42
ATP1A4 Q13733 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ABCB11 O95342 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29382857 0.80 AGXT (0.66) AGXTCYP2C9KMT2AWDR5PDE10A
SCHEMBL1060082 0.80 AGXT (0.66) AGXTCYP2C9KMT2AWDR5PDE10A
Hydrochloric Acid SCHEMBL3247161 0.79 AGXT (0.64) AGXTCYP2C9KMT2AWDR5PDE10A
SCHEMBL17434548 0.79 AGXT (0.64) AGXTCYP2C9KMT2AWDR5PDE10A
SCHEMBL154027 0.77 AGXT (0.66) AGXTCYP2C9KMT2AWDR5PDE10A
SCHEMBL13011461 0.75 AGXT (0.55) AGXTCYP2C9KMT2AWDR5PDE10A
SCHEMBL1160150 0.75 AGXT (0.64) AGXTCYP2C9KMT2AWDR5PDE10A
SCHEMBL22912532 0.75 AGXT (0.74) AGXTCYP2C9KMT2AWDR5PDE10A
SCHEMBL1056427 0.75 AGXT (0.69) AGXTCYP2C9KMT2AWDR5PDE10A
SCHEMBL30209599 0.75 AGXT (0.64) AGXTCYP2C9KMT2AWDR5PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8378100-B2 Phosphonate derivatives as autotaxin inhibitors UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2013-02-19 US disclosed
US-20100016258-A1 PHOSPHONATE DERIVATIVES AS AUTOTAXIN INHIBITORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2010-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100016258-A1 PHOSPHONATE DERIVATIVES AS AUTOTAXIN INHIBITORS ENPP2, PHPT1, GNPAT AGXT 77/4885CYP2C9 4835/4885KMT2A 1976/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.