SCHEMBL3800830

SCHEMBL3800830

Fc1cccc(Cl)c1-c1ncc(-c2ccc(-c3ccc(C(F)(F)F)cc3)nc2)[nH]1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGES O14684 7/20 0.54
SCN2A Q99250 5/20 0.49
JAK2 O60674 1/20 0.49
HPGDS O60760 2/20 0.48
NPY5R Q15761 2/20 0.46
TRPV1 Q8NER1 1/20 0.45
KDM4E B2RXH2 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PTGS1 P23219 1/20 0.38
DGAT1 O75907 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076235 0.82 PTGES (0.49) PTGESJAK2KDM4ENPSR1PTGS1
SCHEMBL3794463 0.80 PTGES (0.67) PTGESSCN2AJAK2HPGDS
SCHEMBL3795117 0.78 PTGES (0.54) PTGESJAK2HPGDSNPY5RKDM4E
SCHEMBL3791357 0.77 PTGES (0.56) PTGESSCN2AJAK2HPGDSNPY5R
SCHEMBL3797909 0.77 PTGES (0.51) PTGESJAK2HPGDS
SCHEMBL3790651 0.77 PTGES (0.51) PTGESJAK2HPGDSNPY5RNPSR1
SCHEMBL3793877 0.76 PTGES (0.55) PTGESSCN2AJAK2HPGDSKDM4E
SCHEMBL3791993 0.76 PTGES (0.50) PTGESJAK2HPGDSNPY5R
SCHEMBL3790517 0.75 PTGES (0.54) PTGESSCN2AJAK2HPGDSKDM4E
SCHEMBL3792008 0.75 PTGES (0.62) PTGESSCN2AJAK2HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed