SCHEMBL3801441

SCHEMBL3801441

O=C(O)c1[nH]c(-c2c(F)cccc2Cl)nc1-c1ccc(C#Cc2ccccc2)nc1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGES O14684 19/20 0.75
GRM5 P41594 1/20 0.38
JAK2 O60674 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3791390 0.93 PTGES (0.72) PTGESGRM5
SCHEMBL13075498 0.90 PTGES (0.69) PTGESGRM5
SCHEMBL3794464 0.88 PTGES (0.66) PTGES
SCHEMBL13076377 0.85 PTGES (0.79) PTGESJAK2
SCHEMBL3795330 0.85 PTGES (1.00) PTGESJAK2
SCHEMBL3795999 0.85 PTGES (0.66) PTGESGRM5JAK2
SCHEMBL3793316 0.84 PTGES (0.76) PTGESJAK2
SCHEMBL13075518 0.83 PTGES (0.51) PTGESJAK2
SCHEMBL3717114 0.81 PTGES (0.64) PTGESGRM5JAK2
SCHEMBL3796674 0.80 PTGES (0.67) PTGESGRM5JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed