SCHEMBL3811248

SCHEMBL3811248

CC(c1ccc(-c2ccc(F)cc2F)cc1)N1CCC(CCOP(=O)(O)O)(c2ccc(F)cc2)OC1=O

nearest known ligand 0.79

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 20/20 0.79
CYP3A4 P08684 9/20 0.79
CYP2C9 P11712 4/20 0.79
CYP2C19 P33261 3/20 0.79
HSD3B2 P26439 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL958981 1.00 HSD11B1 (0.79) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL958979 1.00 HSD11B1 (0.79) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL955842 0.91 HSD11B1 (0.82) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL955840 0.91 HSD11B1 (0.82) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL958995 0.91 HSD11B1 (0.80) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL958996 0.91 HSD11B1 (0.80) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL958994 0.91 HSD11B1 (0.80) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL957665 0.89 HSD11B1 (0.84) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL957664 0.89 HSD11B1 (0.84) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2
SCHEMBL960361 0.88 HSD11B1 (1.00) HSD11B1CYP3A4CYP2C9CYP2C19HSD3B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183228-A1 CYCLIC INHIBITORS OF 11ß -HYDROXYSTERIOD DEHYDROGENASE 1 Vitae Pharmaceuticals, Inc. (US) 2010-05-12 EP claimed
WO-2009017664-A1 CYCLIC INHIBITORS OF 11β-HYDROXYSTERIOD DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-02-05 WO claimed