SCHEMBL3812410

SCHEMBL3812410

CC(C)N1CCN(Cc2ccc(-c3cnc(CN)c(-c4ccnc(-c5ccn(C)n5)c4)c3)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.40
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
TGFBR1 P36897 3/20 0.38
ACVR1 Q04771 3/20 0.38
JMJD6 Q6NYC1 1/20 0.37
TNIK Q9UKE5 5/20 0.36
MAP3K11 Q16584 2/20 0.36
PIK3CA P42336 3/20 0.36
PIK3CD O00329 2/20 0.36
PIK3R1 P27986 2/20 0.36
PIK3CB P42338 2/20 0.36
PIK3CG P48736 2/20 0.36
CDK1 P06493 1/20 0.36
CDK4 P11802 1/20 0.36
CCNB1 P14635 1/20 0.36
CCND1 P24385 1/20 0.36
CDK6 Q00534 1/20 0.36
MAP4K1 Q92918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4186047 0.77 PARP1 (0.41) LRRK2PARP1PARP2ACVR1PIK3CA
SCHEMBL3726227 0.72 PARP1 (0.39) PARP1PARP2ACVR1PIK3CAPIK3CD
SCHEMBL25833013 0.68 SCN4A (0.45) LRRK2
SCHEMBL3717465 0.67 DRD2 (0.41) PARP1PARP2TGFBR1ACVR1PIK3CA
SCHEMBL3659202 0.66 ABL1 (0.45) PARP1PARP2TGFBR1PIK3CAPIK3CD
SCHEMBL3717439 0.65 DRD2 (0.42) LRRK2PARP1PARP2TGFBR1ACVR1
SCHEMBL13743307 0.65 PIK3CD (0.46) PARP1PARP2TGFBR1ACVR1PIK3CA
SCHEMBL3662134 0.64 PIK3CD (0.45) PARP1PARP2PIK3CAPIK3CDPIK3R1
SCHEMBL3066932 0.64 HRH3 (0.57)
SCHEMBL3057408 0.63 CDK6 (0.49) PARP1PARP2CDK1CDK4CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2242742-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2010-10-27 EP disclosed
WO-2009087212-A2 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 2009-07-16 WO disclosed