SCHEMBL3812593

SCHEMBL3812593

Cc1ccc(-c2cc(C(=O)NC(C)c3noc(C)n3)cc(-c3ncccc3F)c2)nc1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 12/20 0.69
P2RX2 Q9UBL9 11/20 0.69
NR1I2 O75469 3/20 0.69
CYP2C9 P11712 2/20 0.47
UGT1A1 P22309 1/20 0.47
MET P08581 1/20 0.41
DGAT2 Q96PD7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3061491 1.00 P2RX3 (0.69) P2RX3P2RX2NR1I2CYP2C9UGT1A1
SCHEMBL2183696 0.82 P2RX3 (0.63) P2RX3P2RX2NR1I2CYP2C9UGT1A1
SCHEMBL21091896 0.82 P2RX3 (0.56) P2RX3P2RX2NR1I2
SCHEMBL3063281 0.81 P2RX3 (1.00) P2RX3P2RX2NR1I2CYP2C9UGT1A1
SCHEMBL13095503 0.80 NR1I2 (0.50) P2RX3P2RX2NR1I2CYP2C9UGT1A1
SCHEMBL3057997 0.76 P2RX3 (0.63) P2RX3P2RX2NR1I2CYP2C9UGT1A1
SCHEMBL3064190 0.75 P2RX3 (0.62) P2RX3P2RX2NR1I2CYP2C9UGT1A1
SCHEMBL13095460 0.75 NR1I2 (0.47) P2RX3P2RX2NR1I2CYP2C9UGT1A1
SCHEMBL13092766 0.74 NR1I2 (0.48) P2RX3P2RX2NR1I2CYP2C9UGT1A1
SCHEMBL3068648 0.72 P2RX3 (0.50) P2RX3P2RX2NR1I2CYP2C9UGT1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215049-A1 P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN Merck Sharp & Dohme Corp. (US) 2010-08-11 EP claimed
WO-2009058298-A1 P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN MERCK & CO., INC. (US) 2009-05-07 WO claimed