SCHEMBL3813652

SCHEMBL3813652

C1CCC(NC2CCNC2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.57
HSD17B10 Q99714 1/20 0.57
EPHX1 P07099 2/20 0.47
KCNH2 Q12809 1/20 0.45
KDM1A O60341 4/20 0.41
MAOB P27338 3/20 0.41
MAOA P21397 1/20 0.41
ADH1B P00325 2/20 0.36
ADH1C P00326 2/20 0.36
ADH1A P07327 2/20 0.36
ADH4 P08319 1/20 0.36
RAD52 P43351 1/20 0.33
GNAI3 P08754 1/20 0.33
GNAO1 P09471 1/20 0.33
GNAI1 P63096 1/20 0.33
ADH7 P40394 1/20 0.32
CISD1 Q9NZ45 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR1B P28222 1/20 0.32
HTR2A P28223 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5827271 1.00 ALDH1A1 (0.57) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
SCHEMBL2878079 0.98 ALDH1A1 (0.52) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
SCHEMBL2877988 0.98 ALDH1A1 (0.52) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
SCHEMBL2877987 0.98 ALDH1A1 (0.52) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
Hydrochloric Acid SCHEMBL2868834 0.95 ALDH1A1 (0.50) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
Hydrochloric Acid SCHEMBL2868836 0.95 ALDH1A1 (0.50) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
Hydrochloric Acid SCHEMBL2875182 0.95 ALDH1A1 (0.50) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
SCHEMBL21425605 0.93 KCNH2 (0.46) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
SCHEMBL5808030 0.93 KCNH2 (0.46) ALDH1A1HSD17B10EPHX1KCNH2KDM1A
Hydrochloric Acid SCHEMBL31209185 0.91 KCNH2 (0.45) ALDH1A1HSD17B10EPHX1KCNH2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2582692-B1 CYCLOHEXYL-AZETIDINYL ANTAGONISTS OF CCR2 JANSSEN PHARMACEUTICA NV (BE) 2015-07-22 EP disclosed
EP-2089354-A1 NAPHTHALENYLOXYPROPENYL DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME Korea Research Institute Of Chemical Technology (KR) 2009-08-19 EP disclosed
WO-2008054154-A1 NAPHTHALENYLOXYPROPENYL DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2008-05-08 WO disclosed
US-7049323-B2 Amidoheterocycles as modulators of the melanocortin-4 receptor BRISTOL-MYERS SQUIBB COMPANY (US) 2006-05-23 US disclosed
US-20040224901-A1 Amidoheterocycles as modulators of the melanocortin-4 receptor BRISTOL-MYERS SQUIBB COMPANY 2004-11-11 US disclosed
EP-0105665-B1 AZLACTONE-FUNCTIONAL COMPOUNDS AND CURABLE COMPOSITIONS CONTAINING SAME MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1987-12-02 EP disclosed
US-4639286-A Curable compositions containing azlactone-functional compounds MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1987-01-27 US disclosed
US-4485236-A NUCLEOPHILIC GROUP SUBSTITUTION; CROSSLINKED POLYAMIDE RESIN SYSTEMS MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1984-11-27 US disclosed
EP-0105665-A1 Azlactone-functional compounds and curable compositions containing same MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1984-04-18 EP disclosed
US-4005208-A GASTRIC JUICE, ANTISECRETORY SMITHKLINE CORPORATION (US) 1977-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040224901-A1 Amidoheterocycles as modulators of the melanocortin-4 receptor MC4R, MC1R, MC3R ALDH1A1 4095/4885HSD17B10 1532/4885EPHX1 3709/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.