SCHEMBL381490

SCHEMBL381490

CC(C)(C)N(C(=O)O)C(CO)c1cccc(Cl)c1F

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CFD P00746 1/20 0.40
CXCL8 P10145 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
NOTUM Q6P988 1/20 0.33
OPRM1 P35372 2/20 0.32
MRGPRX4 Q96LA9 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CTSA P10619 1/20 0.31
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16504458 0.90 CFD (0.41) CFDCXCL8NOTUMOPRM1CTSA
SCHEMBL16504457 0.90 CFD (0.41) CFDCXCL8NOTUMOPRM1CTSA
SCHEMBL19244855 0.86 MEN1 (0.41) CXCL8OPRM1MEN1KMT2A
SCHEMBL382379 0.86 NISCH (0.43) CXCL8OPRM1ADRB2ADRB1
SCHEMBL16504550 0.86 CFD (0.40) CFDCXCL8NOTUMOPRM1MRGPRX4
SCHEMBL16504549 0.86 CFD (0.40) CFDCXCL8NOTUMOPRM1MRGPRX4
SCHEMBL15772238 0.78 CFD (0.36) CFDCXCL8SLC6A2SLC6A4SLC6A3
SCHEMBL15772237 0.78 CFD (0.36) CFDCXCL8SLC6A2SLC6A4SLC6A3
SCHEMBL381228 0.76 MEN1 (0.39) CXCL8OPRM1MEN1KMT2A
SCHEMBL382428 0.76 ACP3 (0.43) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408751-B1 Substituted 2-acetamido-5-aryl-1,2,4-triazolones and use thereof BAYER IP GMBH (DE) 2017-08-23 EP disclosed
EP-2408751-A1 Substituted 2-acetamido-5-aryl-1,2,4-triazolones and use thereof Bayer Pharma Aktiengesellschaft (DE) 2012-01-25 EP disclosed
WO-2010105770-A1 SUBSTITUTED 2-ACETAMIDO-5-ARYL-1,2,4-TRIAZOLONES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-09-23 WO disclosed