SCHEMBL3814930

SCHEMBL3814930

COCCOc1cccc(N)c1S(=O)(=O)Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
ALDH1A1 P00352 4/20 0.36
ADRA2B P18089 1/20 0.35
PTGS1 P23219 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
FFAR2 O15552 1/20 0.35
EGFR P00533 2/20 0.34
L3MBTL1 Q9Y468 4/20 0.33
POLB P06746 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
RECQL P46063 1/20 0.33
IKBKB O14920 1/20 0.33
TIPARP Q7Z3E1 1/20 0.33
KDM1A O60341 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763665 0.82 ALDH1A1 (0.50) ALDH1A1ADRA2BPTGS1TDP1POLB
SCHEMBL3824646 0.77 CYP3A4 (0.40) ALDH1A1ADRA2BL3MBTL1LMNAGAA
SCHEMBL8136765 0.77 CYP1A2 (0.44) CYP1A2CYP2C9CYP2C19HDAC3HDAC1
SCHEMBL2846218 0.76 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19HDAC3HDAC1
SCHEMBL31172404 0.76 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19HDAC3HDAC1
SCHEMBL29684634 0.76 CYP1A2 (0.66) CYP1A2CYP2C9CYP2C19HDAC3HDAC1
SCHEMBL1029928 0.76 CYP1A2 (0.66) CYP1A2CYP2C9CYP2C19HDAC3HDAC1
SCHEMBL23352277 0.75 CYP1A2 (0.44) CYP1A2CYP2C9CYP2C19KDM4ELMNA
SCHEMBL13537676 0.73 CYP1A2 (0.44) CYP1A2CYP2C9CYP2C19HDAC3HDAC1
SCHEMBL10812034 0.73 ADORA2A (0.51) CYP1A2CYP2C9CYP2C19ALDH1A1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009141065-A2 (1,2-BENZISOTHIAZOL-3-YL)(THIO)CARBAMATES AND (1,2-BENZISOTHIAZOL-3-YL)(THIO)OXAMATES AND THE OXIDATION FORMS THEREOF FOR USE AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2009-11-26 WO disclosed
EP-2123159-A1 (1,2-Benzisothiazol-3-yl)(thio)carbamates and (1,2-Benzisothiazol-3-yl)(thio)oxamates and their oxidation forms as pesticides Bayer CropScience AG (DE) 2009-11-25 EP disclosed