SCHEMBL3818352

SCHEMBL3818352

O=C1O[C@@H](CO)CN1c1ccc(OC[C@H]2CCNC2)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CALML3 P27482 6/20 0.51
MAOA P21397 6/20 0.46
MAOB P27338 3/20 0.44
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP3A4 P08684 1/20 0.42
TLR9 Q9NR96 1/20 0.41
TLR8 Q9NR97 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
F10 P00742 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL542051 1.00 CALML3 (0.51) CALML3MAOAMAOBCYP2C19CYP2C9
SCHEMBL541746 0.95 CALML3 (0.53) CALML3MAOAMAOBCYP2C19CYP2C9
SCHEMBL541747 0.95 CALML3 (0.53) CALML3MAOAMAOBCYP2C19CYP2C9
SCHEMBL10033726 0.87 MAOA (0.56) CALML3MAOAMAOBF10
SCHEMBL10066190 0.87 MAOA (0.56) CALML3MAOAMAOBF10
SCHEMBL10033727 0.87 MAOA (0.56) CALML3MAOAMAOBF10
SCHEMBL10033721 0.83 MAOA (0.57) CALML3MAOAMAOBF10
SCHEMBL542046 0.80 CALML3 (0.53) CALML3MAOAMAOBCYP2C19CYP2C9
SCHEMBL542047 0.80 CALML3 (0.53) CALML3MAOAMAOBCYP2C19CYP2C9
SCHEMBL10033753 0.80 MAOA (0.54) CALML3MAOAMAOBF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2086968-A1 5-HYDROXYMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-08-12 EP disclosed
WO-2008056335-A1 5-HYDROXYMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-05-15 WO disclosed