SCHEMBL3819964

SCHEMBL3819964

Cc1cc(C)c2oc(Nc3ccc(-c4nn(C5CCC(N6CCNC(=O)C6)CC5)c5ncnc(N)c45)cc3F)nc2c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.78
IGF1R P08069 16/20 0.78
ERBB4 Q15303 15/20 0.78
ERBB2 P04626 14/20 0.78
ERBB3 P21860 14/20 0.78
AURKB Q96GD4 5/20 0.61
AURKA O14965 4/20 0.61
PLK4 O00444 2/20 0.55
MAPK13 O15264 2/20 0.55
PDPK1 O15530 2/20 0.55
DAPK3 O43293 2/20 0.55
JAK2 O60674 2/20 0.55
ROCK2 O75116 2/20 0.55
PAK4 O96013 2/20 0.55
ABL1 P00519 2/20 0.55
NTRK1 P04629 2/20 0.55
INSR P06213 2/20 0.55
LCK P06239 2/20 0.55
FYN P06241 2/20 0.55
CDK1 P06493 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6108400 1.00 EGFR (0.78) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL4820117 0.91 IGF1R (0.67) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL4820107 0.91 IGF1R (0.67) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL4824623 0.91 IGF1R (0.67) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL6430800 0.88 EGFR (1.00) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL4819751 0.88 EGFR (1.00) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL6109791 0.82 EGFR (0.73) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL6109795 0.82 EGFR (0.73) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL3830176 0.81 EGFR (0.72) EGFRIGF1RERBB4ERBB2ERBB3
SCHEMBL4824147 0.81 EGFR (0.63) EGFRIGF1RERBB4ERBB2ERBB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730148-A4 AMINOBENZOXAZOLES AS THERAPEUTIC AGENTS ABBOTT LAB (US) 2009-08-19 EP disclosed
EP-1730148-A2 AMINOBENZOXAZOLES AS THERAPEUTIC AGENTS Abbott Laboratories (US) 2006-12-13 EP disclosed
US-20060025383-A1 Aminobenzoxazoles as therapeutic agents ABBOTT LABORATORIES 2006-02-02 US disclosed
WO-2005074603-A2 AMINOBENZOXAZOLES AS THERAPEUTIC AGENTS ABBOTT LABORATORIES (US) 2005-08-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060025383-A1 Aminobenzoxazoles as therapeutic agents ABL1, MAP3K19, MAP3K20 EGFR 506/4885IGF1R 2859/4885ERBB4 157/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.