SCHEMBL3820604

SCHEMBL3820604

CC(C)CN(c1ccc(C#N)c(Cl)c1)[C@H]1CCN(C(=O)C(C)C)C1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PGR P06401 20/20 0.71
CYP2C9 P11712 20/20 0.71
CYP2D6 P10635 18/20 0.71
KCNH2 Q12809 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3820608 1.00 PGR (0.71) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162171 0.93 PGR (0.70) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3822700 0.91 PGR (0.62) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3827209 0.88 PGR (0.68) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3827821 0.88 PGR (0.68) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3842491 0.85 PGR (0.81) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3826345 0.85 PGR (0.90) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3842487 0.85 PGR (0.81) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3029850 0.83 PGR (0.78) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162332 0.83 PGR (0.61) PGRCYP2C9CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094269-A1 PYRROLIDINANILINES Smithkline Beecham Corporation (US) 2009-09-02 EP disclosed
WO-2008077089-A1 PYRROLIDINANILINES SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed