SCHEMBL382125

SCHEMBL382125

COc1cc(N2CCNCC2)ccc1Nc1ncc(Cl)c(NCc2ccccc2S(N)(=O)=O)n1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.69
ALK Q9UM73 8/20 0.68
JAK2 O60674 1/20 0.58
SRC P12931 1/20 0.58
TNK2 Q07912 1/20 0.58
ZAP70 P43403 2/20 0.57
IGF1R P08069 1/20 0.55
KCNH2 Q12809 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382126 0.84 EGFR (0.70) EGFRALKZAP70IGF1R
SCHEMBL10205065 0.82 ALK (0.64) EGFRALKJAK2SRCTNK2
SCHEMBL21846989 0.82 EGFR (1.00) EGFRALK
SCHEMBL382124 0.81 ALK (0.81) EGFRALKZAP70IGF1R
SCHEMBL16752958 0.81 ALK (1.00) EGFRALK
SCHEMBL26161575 0.80 ALK (0.85) EGFRALKIGF1RKCNH2
SCHEMBL21846999 0.80 EGFR (1.00) EGFRALK
SCHEMBL18506895 0.79 ALK (0.66) EGFRALKJAK2IGF1RKCNH2
SCHEMBL30502344 0.79 ALK (0.87) EGFRALKIGF1RKCNH2
SCHEMBL29188606 0.78 ALK (0.82) EGFRALKIGF1RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1660458-B1 2, 4-PYRIMIDINEDIAMINES USEFUL IN THE TREATMENT OF NEOPLASTIC DISEASES, INFLAMMATORY AND IMMUNE SYSTEM DISORDERS NOVARTIS AG (CH) 2012-01-25 EP disclosed